Target Details
| UniProt AC | Q9UM73 |
|---|---|
| Gene Symbol | ALK |
| Protein Name | ALK tyrosine kinase receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12810 (ALK_LTK_GRD) PF00629 (MAM) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 712
- Clinical molecules 27
- Avg pChEMBL 7.64
KEGG Pathways (3)
Associated Diseases (4)
Active Molecules (712)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XQCYJMDRMXBJIP
|
7.5 | IC50 | 2 | — | |
GMAZSCDBFSDVRI
|
7.5 | IC50 | 3 | — | |
LDRVTAIULYJYRP
|
7.5 | IC50 | 2 | — | |
OUCKZVRLUAQTBL
|
7.5 | IC50 | 3 | — | |
XFABGERDXKXSEQ
|
7.5 | IC50 | 2 | — | |
CHQPVKQIKUZXJB
|
7.5 | IC50 | 2 | — | |
QCNWNKFYASABSV
|
7.5 | IC50 | 2 | — | |
XZXHXSATPCNXJR
|
7.5 | Kd | 165 | Yes | |
AQRHXRWJOUUDKH
|
7.5 | IC50 | 2 | — | |
FAUWHVUDSIQEKF
|
7.5 | IC50 | 3 | — | |
QRCUKJSISICWNH
|
7.5 | IC50 | 2 | — | |
AZXPDNLEMGQMQS
|
7.5 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.5 | Kd | 213 | — | |
HBJCTXQIDBQUKL
|
7.5 | IC50 | 2 | — | |
NBLXWOQTZXCMKV
|
7.5 | IC50 | 3 | — | |
XJKVPKPXYHLAKR
|
7.5 | IC50 | 2 | — | |
FZBVNCFBCNXULH
|
7.5 | IC50 | 18 | — | |
GPJRGBLZCBBYMB
|
7.5 | IC50 | 2 | — | |
HATRKFPXWDUKPL
|
7.5 | IC50 | 3 | — | |
NNWRFTLSEJKLQI
|
7.5 | IC50 | 2 | — | |
PYEVUJXYLLDVLP
|
7.5 | IC50 | 2 | — | |
ICYMRJXTNSDJCF
|
7.4 | IC50 | 2 | — | |
UAVBPSVJXCTZOC
|
7.4 | IC50 | 3 | — | |
UIFHDCIICKTEAL
|
7.4 | IC50 | 3 | — | |
AGEWKUQZNAGGEC
|
7.4 | IC50 | 2 | — | |
ADQFBAMWKUTCQJ
|
7.4 | IC50 | 2 | — | |
GHJLZINDIHSFBZ
|
7.4 | IC50 | 2 | — | |
LUZLOIYOYLEIRH
|
7.4 | IC50 | 2 | — | |
WTLGABJSLMBEHB
|
7.4 | IC50 | 2 | — | |
XYJHFAIWNWCPJD
|
7.4 | IC50 | 2 | — | |
PIRWRQQYRXWTII
|
7.4 | IC50 | 3 | — | |
DSSRVQAIWBZWON
|
7.4 | Ki | 9 | — | |
MQZWITYZSPAJLX
|
7.4 | IC50 | 2 | — | |
BPGJJKMCXBBEBI
|
7.4 | IC50 | 2 | — | |
RCSMIXJVDRCRBA
|
7.4 | IC50 | 2 | — | |
FLTLUXCGVBUQLQ
|
7.4 | IC50 | 3 | — | |
FLTLUXCGVBUQLQ
|
7.4 | IC50 | 3 | — | |
HZUPDOJVKYRRMY
|
7.4 | IC50 | 3 | — | |
PFZIQVWSNDVNQV
|
7.4 | IC50 | 2 | — | |
SVQKJNKAPILWNS
|
7.4 | IC50 | 2 | — | |
AHLIOYKRAKANRB
|
7.4 | IC50 | 2 | — | |
BMDPGNPXJLGRNG
|
7.4 | IC50 | 2 | — | |
OOXXIVRLCXQRPS
|
7.4 | IC50 | 2 | — | |
SOBJVDFONGAIIH
|
7.4 | IC50 | 2 | — | |
UYBILPBKQDAXTL
|
7.4 | IC50 | 2 | — | |
ZKHQZMGFQLTDQH
|
7.4 | IC50 | 3 | — | |
WDFURCPOBHRTIU
|
7.3 | IC50 | 2 | — | |
CTOIWJDYNIQZEG
|
7.3 | IC50 | 2 | — | |
CTZVCMKQQAGWBA
|
7.3 | IC50 | 3 | — | |
MNUHUBSGVGOPGM
|
7.3 | IC50 | 3 | — |