Target Details
| UniProt AC | Q9UM73 |
|---|---|
| Gene Symbol | ALK |
| Protein Name | ALK tyrosine kinase receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12810 (ALK_LTK_GRD) PF00629 (MAM) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 712
- Clinical molecules 27
- Avg pChEMBL 7.64
KEGG Pathways (3)
Associated Diseases (4)
Active Molecules (712)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
INVMLEPLZRDFOO
|
7.7 | IC50 | 2 | — | |
ROGKAFOTXRPAFP
|
7.7 | IC50 | 2 | — | |
TZQJLQWNUAZYJQ
|
7.7 | IC50 | 3 | — | |
CKOFEFWHTQQMLF
|
7.7 | IC50 | 2 | — | |
HSCSBODZXPHWFM
|
7.7 | IC50 | 2 | — | |
IFENGTVBYLDKRT
|
7.7 | IC50 | 2 | — | |
NMJMRSQTDLRCRQ
|
7.7 | IC50 | 7 | — | |
CPVCXTGQEFSNOQ
|
7.7 | IC50 | 2 | — | |
JHZOJILVCGEIFB
|
7.7 | IC50 | 3 | — | |
MTJABDOZWOEWJD
|
7.7 | IC50 | 2 | — | |
FQUQLTHTCSOGBY
|
7.7 | IC50 | 3 | — | |
ITNPURPVZHRALQ
|
7.7 | IC50 | 2 | — | |
IGJYHELICIRMRM
|
7.6 | IC50 | 2 | — | |
NKGBJFZCCPPWIY
|
7.6 | IC50 | 2 | — | |
NXKBBURYGABXCP
|
7.6 | IC50 | 2 | — | |
RKWOVOVDWBRGQO
|
7.6 | IC50 | 5 | — | |
UYIANZRYPSGDFM
|
7.6 | IC50 | 2 | — | |
FGPCDMAFJXAZGK
|
7.6 | IC50 | 2 | — | |
PCAABRMAORWYHN
|
7.6 | IC50 | 2 | — | |
DCQGBFHFVFACQU
|
7.6 | IC50 | 3 | — | |
DRPOUFRDMKUUKI
|
7.6 | IC50 | 2 | — | |
HAGKVAUHAUZMBY
|
7.6 | IC50 | 2 | — | |
IIFZHKOYTWEVOZ
|
7.6 | IC50 | 2 | — | |
WLTMYDRAYRGWMO
|
7.6 | IC50 | 5 | — | |
ADDQRQHBRAHARB
|
7.6 | Ki | 2 | — | |
GLGNXYJARSMNGJ
|
7.6 | IC50 | 2 | — | |
KKYPRNBBPBRJQX
|
7.6 | Ki | 40 | — | |
MFPZJISOIZABEX
|
7.6 | IC50 | 2 | — | |
PIBITIKJRIGPID
|
7.6 | IC50 | 3 | — | |
UYJNQQDJUOUFQJ
|
7.6 | IC50 | 68 | — | |
XJBVBERAWLJSDE
|
7.6 | IC50 | 2 | — | |
XKFTZKGMDDZMJI
|
7.6 | Ki | 56 | — | |
ADAQBVKANMBBGO
|
7.6 | IC50 | 2 | — | |
QGVMEYLFVOBUHE
|
7.6 | IC50 | 2 | — | |
RZSXKXZMLBUVEC
|
7.6 | IC50 | 2 | — | |
LOLWMDGFTABZFN
|
7.6 | IC50 | 2 | — | |
VYUPBBUIPPRDHY
|
7.6 | IC50 | 4 | — | |
YKKQUJHYJQWYHQ
|
7.6 | IC50 | 3 | — | |
ARFSIMCXZSKBGL
|
7.6 | IC50 | 3 | — | |
FGRVKMDGFGXLDX
|
7.6 | IC50 | 5 | — | |
HKTKCWHAQWAVOW
|
7.6 | IC50 | 5 | — | |
MPLLJMUCCXFTPL
|
7.6 | IC50 | 3 | — | |
OUBJSHKDVMRZQJ
|
7.6 | IC50 | 5 | — | |
SCHLJLHHIALWBK
|
7.6 | IC50 | 5 | — | |
XNLDXKJZCGYOAU
|
7.6 | IC50 | 5 | — | |
ZCIQMENOTTVELZ
|
7.6 | IC50 | 3 | — | |
AMSONZZHZCNUHV
|
7.5 | IC50 | 2 | — | |
DCMKAPVKXJVEOA
|
7.5 | IC50 | 2 | — | |
MVLCLEZORCBEHN
|
7.5 | Kd | 2 | — | |
WAGRWRIWWPGPDN
|
7.5 | IC50 | 2 | — |