Target Details
| UniProt AC | Q9UM73 |
|---|---|
| Gene Symbol | ALK |
| Protein Name | ALK tyrosine kinase receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12810 (ALK_LTK_GRD) PF00629 (MAM) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 712
- Clinical molecules 27
- Avg pChEMBL 7.64
KEGG Pathways (3)
Associated Diseases (4)
Active Molecules (712)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HQZLQPMNIPRNBQ
|
7.8 | IC50 | 3 | — | |
KXPICMSXZCNILY
|
7.8 | IC50 | 2 | — | |
MFUMJAGTBAKMKI
|
7.8 | IC50 | 2 | — | |
MTZNLMGFYVEIAP
|
7.8 | IC50 | 2 | — | |
MVMGHPHRNLHXAW
|
7.8 | IC50 | 2 | — | |
ZIPMVFDKNBGKAT
|
7.8 | IC50 | 3 | — | |
PURNBEBZVYETFI
|
7.8 | IC50 | 3 | — | |
COZPORUDEQRJMN
|
7.8 | IC50 | 3 | — | |
JVCFOBYUGHIPJO
|
7.8 | IC50 | 2 | — | |
MBDRYJSNQAFOKD
|
7.8 | IC50 | 2 | — | |
OVRQGEYZDUHJNZ
|
7.8 | IC50 | 2 | — | |
OWFXKTOLFUQPDJ
|
7.8 | Ki | 36 | — | |
PUPCRRRSBUYJAD
|
7.8 | Ki | 44 | Yes | |
YEFKWCQOENUXOA
|
7.8 | IC50 | 2 | — | |
COCRBNKPTJZHDN
|
7.8 | IC50 | 2 | — | |
ILSYFQQNAQIMBK
|
7.8 | IC50 | 2 | — | |
LMBKLNFIUZRASR
|
7.8 | IC50 | 2 | — | |
RLDIJFHXXAQFAJ
|
7.8 | IC50 | 2 | — | |
BCSHRERPHLTPEE
|
7.8 | IC50 | 3 | — | |
CNQREVSEDFUJPZ
|
7.8 | IC50 | 2 | — | |
DUETYWKLKOISFN
|
7.8 | IC50 | 2 | — | |
HVQXOMBEMKJVOC
|
7.8 | IC50 | 2 | — | |
LGIBDQRYOFBMTC
|
7.8 | Ki | 6 | Yes | |
MLXUDJPUEMLBKJ
|
7.8 | IC50 | 2 | — | |
PWAFPCCSKIOXHE
|
7.8 | IC50 | 3 | — | |
CFKDUEIETGGIRT
|
7.8 | IC50 | 2 | — | |
FQUQLTHTCSOGBY
|
7.8 | IC50 | 3 | — | |
JQMFATNHUYQNBF
|
7.8 | IC50 | 2 | — | |
KZXIZEAAKHQALQ
|
7.8 | IC50 | 2 | — | |
OKCOQQXHDZUFTL
|
7.8 | IC50 | 2 | — | |
SOAVEOJCKVRROO
|
7.8 | IC50 | 2 | — | |
ACYSIZUFQATBIE
|
7.8 | IC50 | 2 | — | |
CXFLFTVIZRBMKT
|
7.7 | IC50 | 2 | — | |
FWFBPWPSNFCBOI
|
7.7 | IC50 | 2 | — | |
GDRLJBDXWDATLA
|
7.7 | IC50 | 13 | — | |
QDOTUHIGOCRMSM
|
7.7 | IC50 | 3 | — | |
RPKOZPSDQJWXMG
|
7.7 | IC50 | 2 | — | |
YNWRFXIHAOGUAM
|
7.7 | IC50 | 2 | — | |
ATOVGFGJTVTJSL
|
7.7 | IC50 | 2 | — | |
DPQSQXGBMAXUAP
|
7.7 | IC50 | 3 | — | |
GCVRKWYNRILXKN
|
7.7 | IC50 | 2 | — | |
HCQWDCIGBDDWLZ
|
7.7 | IC50 | 3 | — | |
MOAIIOFZEWYTIP
|
7.7 | IC50 | 3 | — | |
SYZCXHIZVIOJHP
|
7.7 | IC50 | 2 | — | |
UDOCNBYJBDSRQS
|
7.7 | IC50 | 2 | — | |
WUOOWFKJQHKXHK
|
7.7 | IC50 | 4 | — | |
AFTBNZZMNUUEFO
|
7.7 | IC50 | 7 | — | |
FXEXWMOKUBELTG
|
7.7 | IC50 | 2 | — | |
NJPLUFOJYZAGOK
|
7.7 | IC50 | 2 | — | |
QXOZRBMOILEYGU
|
7.7 | IC50 | 2 | — |