Target Details
| UniProt AC | Q9UM73 |
|---|---|
| Gene Symbol | ALK |
| Protein Name | ALK tyrosine kinase receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12810 (ALK_LTK_GRD) PF00629 (MAM) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 712
- Clinical molecules 27
- Avg pChEMBL 7.64
KEGG Pathways (3)
Associated Diseases (4)
Active Molecules (712)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QONPPIZSNSSCSK
|
8.4 | Ki | 45 | Yes | |
QQWUGDVOUVUTOY
|
8.4 | IC50 | 231 | Yes | |
RACYTTCRBPEXAP
|
8.4 | IC50 | 2 | — | |
WXMYXQYBHNGGNH
|
8.4 | IC50 | 2 | — | |
KAALIBYKULTZPV
|
8.4 | IC50 | 2 | — | |
MLJKSWPNIQXPCX
|
8.4 | IC50 | 2 | — | |
IZUHPEAVOSEXHO
|
8.4 | IC50 | 2 | — | |
LVBJEZPSLPIGDT
|
8.4 | IC50 | 2 | — | |
VALNJAQHJPYEAK
|
8.4 | IC50 | 3 | — | |
SFPSNTOXJBCKGE
|
8.4 | IC50 | 2 | — | |
CMVRVFZXCSVCKY
|
8.3 | IC50 | 2 | — | |
ZGFXRISUXOJOLE
|
8.3 | IC50 | 2 | — | |
JKEFKVZKYKUDGL
|
8.3 | IC50 | 2 | — | |
PRUWBPAGUCKXMV
|
8.3 | IC50 | 2 | — | |
DIWRJVJHXXZINL
|
8.3 | IC50 | 4 | — | |
IHRFTDHYCNWNFR
|
8.3 | IC50 | 3 | — | |
BLQJPEQBTMZVKM
|
8.3 | IC50 | 2 | — | |
FCKKFYWNFKXOIH
|
8.3 | IC50 | 2 | — | |
IDGLCVJYKNDJCG
|
8.3 | IC50 | 2 | — | |
IKENQUDOTQBCJH
|
8.3 | IC50 | 18 | — | |
PEKQRSRFUKHNAB
|
8.3 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
8.3 | Ki | 118 | — | |
MOENETCLMCOREY
|
8.3 | IC50 | 2 | — | |
IXBQYIJFDYAVJA
|
8.3 | IC50 | 2 | — | |
JWHAROIQSCGUPR
|
8.3 | IC50 | 2 | — | |
KUFBKQQDUMDVPE
|
8.3 | IC50 | 2 | — | |
CWQBEWYRKVPJHU
|
8.3 | IC50 | 2 | — | |
WTEVQSAOHYKUTI
|
8.3 | IC50 | 2 | — | |
XJPVLMZNDIDZRP
|
8.3 | IC50 | 2 | — | |
GYPCQEWODOUOAU
|
8.3 | IC50 | 2 | — | |
RJLMIOROTJPHHU
|
8.3 | IC50 | 2 | — | |
ATUIHXRIJCYLPA
|
8.3 | IC50 | 4 | — | |
IIXWYSCJSQVBQM
|
8.3 | IC50 | 18 | — | |
LCCBBQQRBMWQEO
|
8.3 | IC50 | 2 | — | |
NHEOMGKMIVQQIX
|
8.3 | IC50 | 4 | — | |
WYRLDZNQPSAQEB
|
8.3 | IC50 | 2 | — | |
LOONVQWRKJLEEG
|
8.2 | IC50 | 8 | — | |
UGWBYFCYZUIYGV
|
8.2 | IC50 | 2 | — | |
SBEYSILWLYDNSN
|
8.2 | IC50 | 2 | — | |
VKTZTNPHNQXFTQ
|
8.2 | IC50 | 4 | — | |
AKHXBNQXYOJHSZ
|
8.2 | IC50 | 2 | — | |
SAHMNRNXZPYQHB
|
8.2 | IC50 | 3 | — | |
BAKDYDIANXRUHQ
|
8.2 | IC50 | 3 | — | |
GYQWOGHOBIBGDV
|
8.2 | IC50 | 4 | — | |
LAJAFFLJAJMYLK
|
8.2 | IC50 | 17 | — | |
JZCIRSHLQAWPRJ
|
8.2 | IC50 | 2 | — | |
KZNWRBSYSUFFOG
|
8.2 | IC50 | 2 | — | |
HVIJVFYUUAELBN
|
8.2 | IC50 | 2 | — | |
PKMJFPBKTISKAX
|
8.2 | IC50 | 3 | — | |
ZFESQIANWCIUCE
|
8.2 | IC50 | 2 | — |