Target Details
| UniProt AC | Q9UM73 |
|---|---|
| Gene Symbol | ALK |
| Protein Name | ALK tyrosine kinase receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12810 (ALK_LTK_GRD) PF00629 (MAM) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 712
- Clinical molecules 27
- Avg pChEMBL 7.64
KEGG Pathways (3)
Associated Diseases (4)
Active Molecules (712)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HVZHUYCJAOSSBB
|
8.6 | IC50 | 2 | — | |
KHNKMLQHLHWWSI
|
8.6 | IC50 | 3 | — | |
STKCTXOVMCUJSB
|
8.6 | IC50 | 4 | — | |
VGPUSZSVCBVTBJ
|
8.6 | IC50 | 2 | — | |
MZGDIKYASHMRSG
|
8.6 | IC50 | 2 | — | |
RBYNLDMNBXNZMS
|
8.6 | IC50 | 4 | — | |
VUPKYIDSZYTBHB
|
8.6 | IC50 | 2 | — | |
WQLHYGLQUAJXEC
|
8.6 | IC50 | 2 | — | |
BDVGHJLTQZVVPA
|
8.6 | IC50 | 2 | — | |
GUUUIDZRGJYTMH
|
8.6 | IC50 | 2 | — | |
MMJWRPJCZSSSNA
|
8.6 | IC50 | 2 | — | |
OIYDABDXSYUHNK
|
8.6 | IC50 | 2 | — | |
SXTUUDANYSHGTB
|
8.6 | IC50 | 2 | — | |
ZJDFSKSBQBPOSK
|
8.6 | IC50 | 24 | Yes | |
ORFGUEWOGJKLFU
|
8.6 | IC50 | 2 | — | |
IVWSMDDTFYCVFZ
|
8.6 | IC50 | 2 | — | |
RWASATDZTQIHPA
|
8.6 | IC50 | 2 | — | |
LTIMJKHVDDEVSP
|
8.5 | IC50 | 2 | — | |
XDTMZEAHVJVNJG
|
8.5 | IC50 | 2 | — | |
QDJZMRPVQLAGDJ
|
8.5 | IC50 | 2 | — | |
TWFGYFUYNRUBKC
|
8.5 | IC50 | 2 | — | |
AOXIGKGAMMGXCX
|
8.5 | IC50 | 2 | — | |
GZSOMRIONXRGEX
|
8.5 | IC50 | 4 | — | |
HKSZLNNOFSGOKW
|
8.5 | IC50 | 408 | — | |
IROGUEMYXINLOZ
|
8.5 | IC50 | 3 | — | |
MYBIYOGYGXIDJG
|
8.5 | IC50 | 2 | — | |
OVDSPTSBIQCAIN
|
8.5 | IC50 | 7 | — | |
SKXAZUOZHANICG
|
8.5 | IC50 | 3 | — | |
XLCWUIJQDPUYAW
|
8.5 | IC50 | 2 | — | |
ZNLXCLMQEIQSAS
|
8.5 | IC50 | 2 | — | |
SXWCURZBDVOHEJ
|
8.5 | IC50 | 2 | — | |
VJWLMBVALMQEMA
|
8.5 | IC50 | 3 | — | |
ZWDPQPKCKRVHBW
|
8.5 | IC50 | 2 | — | |
KYTDVMCLOSUQEH
|
8.5 | IC50 | 2 | — | |
WGEGYCKWUWQOIP
|
8.5 | IC50 | 3 | — | |
BCSHRERPHLTPEE
|
8.5 | IC50 | 3 | — | |
QPNJJRLONMTPQV
|
8.5 | IC50 | 2 | — | |
QOEFDQQUMQBVOB
|
8.5 | IC50 | 2 | — | |
SQPURFIALRFCBJ
|
8.5 | IC50 | 2 | — | |
YLAPHXZIXJJZIH
|
8.5 | IC50 | 2 | — | |
RMBJAPLSOZTGDA
|
8.5 | IC50 | 2 | — | |
SMKJDFHRUWJNRS
|
8.5 | IC50 | 2 | — | |
AJHJEQWEJUXGIF
|
8.4 | IC50 | 4 | — | |
MAKLQLGGXQPLRV
|
8.4 | IC50 | 2 | — | |
XJMFPTCMAYQIDJ
|
8.4 | IC50 | 2 | — | |
FIKPXCOQUIZNHB
|
8.4 | IC50 | 9 | — | |
SNYQSPGQFDKITH
|
8.4 | IC50 | 3 | — | |
VWCZORWQNKCYGE
|
8.4 | IC50 | 17 | — | |
YGYGMNYVMRIARK
|
8.4 | IC50 | 3 | — | |
OWRXHGAFWZFFCW
|
8.4 | Ki | 113 | — |