Target Details
| UniProt AC | Q9UM73 |
|---|---|
| Gene Symbol | ALK |
| Protein Name | ALK tyrosine kinase receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12810 (ALK_LTK_GRD) PF00629 (MAM) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 712
- Clinical molecules 27
- Avg pChEMBL 7.64
KEGG Pathways (3)
Associated Diseases (4)
Active Molecules (712)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HHXONKYVQVDMAS
|
9.0 | IC50 | 3 | — | |
KUKVPUVFVIDHDC
|
9.0 | IC50 | 3 | — | |
MCHOTIIDAJHLED
|
9.0 | IC50 | 5 | Yes | |
UNNQUIYQJKNUQS
|
9.0 | IC50 | 2 | — | |
ADYZVNMLQOHYDE
|
9.0 | IC50 | 2 | — | |
SBLCPBDVMUSESZ
|
9.0 | IC50 | 2 | — | |
SZCXARSUVUOVCP
|
9.0 | IC50 | 3 | — | |
WSTUJEXAPHIEIM
|
9.0 | IC50 | 10 | — | |
HXFVZOYBPSIUHZ
|
8.9 | IC50 | 2 | — | |
RZNBLEUQXRTRGF
|
8.9 | IC50 | 2 | — | |
SSPYHBZSDDTSFN
|
8.9 | IC50 | 9 | — | |
ZCCPLJOKGAACRT
|
8.9 | Kd | 599 | — | |
WHVFDYQCAMPLMS
|
8.9 | Ki | 20 | Yes | |
LEJSTVMXRPKNQA
|
8.9 | IC50 | 2 | — | |
NVHYFDRMQSUXBA
|
8.9 | IC50 | 2 | — | |
IDRQGRCXNROMMS
|
8.9 | IC50 | 3 | — | |
BYWPPTHPCWUJSH
|
8.8 | IC50 | 2 | — | |
DNEAWOPYODVHIL
|
8.8 | IC50 | 2 | — | |
LIBCMUMCEYECFM
|
8.8 | IC50 | 2 | — | |
LLGFEJJPLZCCQL
|
8.8 | IC50 | 10 | Yes | |
UBXWHWZWWVQYGU
|
8.8 | IC50 | 2 | — | |
CENVUXSKJJMKIU
|
8.8 | IC50 | 2 | — | |
RKXGEBJVNGSICG
|
8.8 | IC50 | 3 | — | |
CKZWESXBMQBAAD
|
8.8 | IC50 | 2 | — | |
CSMSPOIEMWPZLD
|
8.8 | IC50 | 2 | — | |
GXWLTJGZFHXMSX
|
8.8 | IC50 | 2 | — | |
HLRNQALVSFYMKM
|
8.8 | IC50 | 3 | — | |
LQLASCOWIMXGMI
|
8.8 | IC50 | 4 | — | |
ZPCCNHQDFZCULN
|
8.8 | IC50 | 2 | — | |
GMAVZOAXIGWUEM
|
8.8 | IC50 | 2 | — | |
AHNSCZJRLJXRAM
|
8.7 | IC50 | 2 | — | |
IXPKKOYDMRELAG
|
8.7 | IC50 | 2 | — | |
SVUZWKKSPKPLEO
|
8.7 | IC50 | 2 | — | |
DRYWSMFQHZVTJK
|
8.7 | IC50 | 3 | — | |
WDRXGELIQZMTRU
|
8.7 | IC50 | 3 | — | |
WUIOBNGTWSVFMF
|
8.7 | IC50 | 2 | — | |
TWJHARJINSWCDD
|
8.7 | IC50 | 2 | — | |
BSZHBKNJHFKROD
|
8.7 | IC50 | 2 | — | |
CQRRHOGDBIREMX
|
8.7 | IC50 | 2 | — | |
FYSRKRZDBHOFAY
|
8.7 | Kd | 8 | — | |
IDGNCVHQDDOPND
|
8.7 | IC50 | 6 | — | |
JJBNBDJXYZZFBC
|
8.7 | IC50 | 3 | — | |
JMSKTSHWCHAIDU
|
8.7 | IC50 | 2 | — | |
LSTKGNJVVPYVIX
|
8.7 | IC50 | 2 | — | |
NFUNPZHOYQJPEH
|
8.7 | IC50 | 2 | — | |
UQWDXRWKSYDDTE
|
8.7 | IC50 | 2 | — | |
UZPCCONBZIFGNY
|
8.7 | IC50 | 2 | — | |
JTUQGTNWWPMBKS
|
8.7 | IC50 | 2 | — | |
QYCCMZVRTHGSBB
|
8.7 | IC50 | 2 | — | |
CAIAMTHZGVFCNA
|
8.6 | IC50 | 2 | — |