Target Details
| UniProt AC | Q9UM73 |
|---|---|
| Gene Symbol | ALK |
| Protein Name | ALK tyrosine kinase receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12810 (ALK_LTK_GRD) PF00629 (MAM) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 712
- Clinical molecules 27
- Avg pChEMBL 7.64
KEGG Pathways (3)
Associated Diseases (4)
Active Molecules (712)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RJTVPQLMBWIFKC
|
6.3 | IC50 | 5 | — | |
XKZINYYXWJEYEL
|
6.3 | Ki | 37 | — | |
ZAARMHXLYCHRAK
|
6.3 | Ki | 20 | — | |
KTEIFNKAUNYNJU
|
6.3 | Kd | 6 | Yes | |
KXMZDGSRSGHMMK
|
6.3 | IC50 | 14 | — | |
AVQNZSIEXOYAGE
|
6.3 | IC50 | 6 | — | |
GUEYLTKEGFGDCH
|
6.2 | IC50 | 4 | — | |
LVXQLMJEKSIZDV
|
6.2 | IC50 | 2 | — | |
FCLVBOUURHAHBG
|
6.2 | IC50 | 2 | — | |
DYUJLNPTOOBZBB
|
6.2 | IC50 | 3 | — | |
QLAIBBCRJCMGRY
|
6.2 | Kd | 2 | — | |
LQNBQZBDXDIOSM
|
6.2 | IC50 | 2 | — | |
AEYLJTAIDDIOBA
|
6.2 | Ki | 53 | — | |
BIIVYFLTOXDAOV
|
6.2 | Ki | 31 | — | |
DZSUJUOJJJCWGG
|
6.2 | Ki | 55 | Yes | |
GCYXEGSPUDSZJY
|
6.2 | Ki | 82 | — | |
JAMDNXUAYUHJLJ
|
6.2 | Ki | 40 | — | |
NVRXTLZYXZNATH
|
6.2 | Ki | 47 | Yes | |
PIQCTGMSNWUMAF
|
6.2 | Ki | 137 | Yes | |
VSVWQTDDGQSGHP
|
6.2 | Ki | 51 | — | |
WDARYLSSWBWVCU
|
6.2 | Ki | 49 | — | |
XJSFDMGICAWQFS
|
6.2 | Ki | 60 | — | |
ZGDYBJXDIXVTLV
|
6.2 | Ki | 54 | — | |
JOOXLOJCABQBSG
|
6.2 | Kd | 139 | — | |
RKGQENOGQBXEPA
|
6.2 | IC50 | 6 | — | |
YYLKKYCXAOBSRM
|
6.2 | Kd | 191 | — | |
BIIVYFLTOXDAOV
|
6.2 | Kd | 29 | — | |
BIIVYFLTOXDAOV
|
6.2 | Kd | 82 | Yes | |
JBNBUAOVEXTUNO
|
6.2 | IC50 | 2 | — | |
WILMKMPUMOSDLH
|
6.2 | IC50 | 5 | — | |
LEHQHFLLRYUONA
|
6.1 | IC50 | 2 | — | |
BETBNWGUKZUUAX
|
6.1 | IC50 | 21 | — | |
QMEZKJBCLUGJTN
|
6.1 | IC50 | 5 | — | |
QMEZKJBCLUGJTN
|
6.1 | IC50 | 4 | — | |
QXPNJMHRUZCEAP
|
6.1 | IC50 | 14 | — | |
KYRYNOGFQDOUCA
|
6.1 | IC50 | 2 | — | |
CHTMRWQLNNRRFJ
|
6.1 | Ki | 70 | — | |
GJKVMXDBPDDFHI
|
6.1 | Ki | 27 | — | |
HXHAJRMTJXHJJZ
|
6.1 | Ki | 52 | Yes | |
JOGKUKXHTYWRGZ
|
6.1 | Ki | 28 | — | |
NFMGZVPRGVERNN
|
6.1 | Ki | 44 | — | |
NXNQLECPAXXYTR
|
6.1 | Ki | 29 | — | |
QLWUDWMYFSWGHK
|
6.1 | Ki | 22 | — | |
GUBJNPWVIUFSTR
|
6.1 | Kd | 103 | — | |
LOGJQOUIVKBFGH
|
6.1 | IC50 | 11 | Yes | |
TULDPDLFHDYJMU
|
6.1 | IC50 | 4 | — | |
BLYRPGBSIKAIAU
|
6.1 | IC50 | 24 | Yes | |
BIKYDWLMTPRSQL
|
6.0 | Ki | 50 | — | |
DJLORVJVWIBDME
|
6.0 | Ki | 24 | — | |
GNLAGGCSJGJECE
|
6.0 | Ki | 19 | Yes |