Target Details
| UniProt AC | Q9UM73 |
|---|---|
| Gene Symbol | ALK |
| Protein Name | ALK tyrosine kinase receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12810 (ALK_LTK_GRD) PF00629 (MAM) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 712
- Clinical molecules 27
- Avg pChEMBL 7.64
KEGG Pathways (3)
Associated Diseases (4)
Active Molecules (712)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BMGQWWVMWDBQGC
|
6.6 | Kd | 147 | Yes | |
PBBXBBSBAJKYLC
|
6.6 | Kd | 3 | — | |
MMZVTNYPOASLID
|
6.6 | IC50 | 3 | — | |
NRFLPOVNIIJIDX
|
6.6 | IC50 | 3 | — | |
NWDUSAJTSMCLKW
|
6.6 | IC50 | 3 | — | |
OEBIHOVSAMBXIB
|
6.6 | IC50 | 5 | — | |
OMVJEQVEBCZADZ
|
6.6 | IC50 | 3 | — | |
PSTULASZQVSGCG
|
6.6 | IC50 | 3 | — | |
SUZGZTADNRRPLU
|
6.6 | IC50 | 3 | — | |
IBAVCNVUPMTBKJ
|
6.5 | IC50 | 5 | — | |
WINJVTFORQNSNW
|
6.5 | IC50 | 2 | — | |
KPXMSUZHJCHOTN
|
6.5 | IC50 | 3 | — | |
WCMQEPUDHFATFM
|
6.5 | IC50 | 3 | — | |
UTNZTKXNTBTXTL
|
6.5 | IC50 | 2 | — | |
ATGVCJYHNOSZEV
|
6.5 | Ki | 23 | — | |
VCFDMLBPASGZTP
|
6.5 | Ki | 38 | — | |
XFWUTMHVDGPWLH
|
6.5 | Ki | 75 | — | |
YEHCNYAQEBQCCS
|
6.5 | Ki | 74 | — | |
YEPNVBNYCRGZRX
|
6.5 | Ki | 26 | — | |
HNIJEISPKOYRAL
|
6.5 | IC50 | 2 | — | |
KQFFSSYWPVJGFN
|
6.5 | IC50 | 2 | — | |
MWVKLRSIDOXBSE
|
6.5 | IC50 | 4 | — | |
FERXSPCVEYOEDT
|
6.5 | IC50 | 4 | — | |
RZRSOLZCLWVUTL
|
6.5 | IC50 | 2 | — | |
WPHKIQPVPYJNAX
|
6.4 | IC50 | 81 | — | |
FERXSPCVEYOEDT
|
6.4 | IC50 | 2 | — | |
JIBBGYSUSKAPDY
|
6.4 | IC50 | 19 | — | |
MIPFBSHTKYTXKN
|
6.4 | IC50 | 2 | — | |
OFUBWOTWQPAEDG
|
6.4 | IC50 | 6 | — | |
WDADYPXHXOFAQY
|
6.4 | IC50 | 2 | — | |
DBBQRLYYNNWGPM
|
6.4 | IC50 | 3 | — | |
AUDNGNGLLRZLDR
|
6.4 | Ki | 33 | — | |
HEUSUIRCBWROMH
|
6.4 | Ki | 64 | — | |
JNAZGEGXKHNDBG
|
6.4 | IC50 | 3 | Yes | |
KOHNRDPXFDZZJF
|
6.4 | Ki | 31 | — | |
LMPULUSZDODHFQ
|
6.4 | Ki | 2 | — | |
LYNBNVBMAGDJRW
|
6.4 | Ki | 81 | — | |
ICYGLDQWNJHCEE
|
6.4 | IC50 | 3 | — | |
MHROCFGPXVNJFS
|
6.4 | IC50 | 3 | — | |
QVDPABSEHBAHOD
|
6.4 | IC50 | 2 | — | |
LYAOPUXRPJKSKW
|
6.4 | IC50 | 3 | — | |
YIKLJNVLVVFHAW
|
6.3 | IC50 | 2 | — | |
CTNPALGJUAXMMC
|
6.3 | Kd | 151 | — | |
NQROQCRXQDNZSD
|
6.3 | IC50 | 3 | — | |
FEQNECCIEFZWKT
|
6.3 | IC50 | 2 | — | |
HFNKQEVNSGCOJV
|
6.3 | Ki | 18 | — | |
KUNZDWIFPOMUOX
|
6.3 | Ki | 36 | — | |
LGHBDVLAHHANMX
|
6.3 | Ki | 53 | — | |
MGNQNQOSSLCUFP
|
6.3 | Ki | 12 | — | |
NOBMKUVHFRVBES
|
6.3 | Ki | 19 | — |