Target Details
| UniProt AC | Q9UM73 |
|---|---|
| Gene Symbol | ALK |
| Protein Name | ALK tyrosine kinase receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12810 (ALK_LTK_GRD) PF00629 (MAM) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 712
- Clinical molecules 27
- Avg pChEMBL 7.64
KEGG Pathways (3)
Associated Diseases (4)
Active Molecules (712)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HUFOZJXAKZVRNJ
|
6.8 | IC50 | 10 | — | |
DYUJLNPTOOBZBB
|
6.8 | IC50 | 3 | — | |
DJORULJHGWXHKA
|
6.8 | IC50 | 2 | — | |
ZHOXAGNPCZTRBN
|
6.8 | Kd | 20 | — | |
ROHJEIACUNTGFP
|
6.8 | IC50 | 16 | — | |
HCNIBOQWDVOZKF
|
6.8 | Ki | 26 | — | |
MULNSLQVKKUPJN
|
6.8 | Ki | 41 | — | |
PYXQMJSGJIJHJT
|
6.8 | Ki | 28 | — | |
VNDWQCSOSCCWIP
|
6.8 | Ki | 39 | Yes | |
WINHZLLDWRZWRT
|
6.8 | Kd | 201 | Yes | |
OSVUGUHRKMMBSE
|
6.8 | Kd | 170 | — | |
YIHUYKCYYKDOHR
|
6.8 | IC50 | 2 | — | |
AEOFEGDYORZHFE
|
6.8 | IC50 | 4 | — | |
DUYJMQONPNNFPI
|
6.8 | IC50 | 11 | — | |
QKYONSSKLFQUAK
|
6.7 | IC50 | 4 | — | |
SRWSLWJKGRZRMC
|
6.7 | Kd | 4 | — | |
UMZFBMAHLWQSBF
|
6.7 | IC50 | 4 | — | |
ZCTFOPDXSRRCIE
|
6.7 | IC50 | 2 | — | |
HFSWCNDZVPIIOF
|
6.7 | IC50 | 8 | — | |
UGPDJIJFANODJH
|
6.7 | IC50 | 12 | — | |
XQVVPGYIWAGRNI
|
6.7 | IC50 | 34 | — | |
YRWVTRIPDNRHAC
|
6.7 | IC50 | 2 | — | |
AXLAIMYZOBLZAF
|
6.7 | IC50 | 2 | — | |
FDVSOQRNTAPCHB
|
6.7 | Ki | 40 | — | |
LODWOBAYUQRWKD
|
6.7 | IC50 | 7 | — | |
MZDKLVOWGIOKTN
|
6.7 | Ki | 80 | — | |
NHFDRBXTEDBWCZ
|
6.7 | Ki | 41 | — | |
NWMPVMMGSHXANZ
|
6.7 | Ki | 58 | — | |
RBXYGQNZRVPDNB
|
6.7 | Ki | 34 | — | |
UBPYILGKFZZVDX
|
6.7 | IC50 | 130 | Yes | |
WUWDLXZGHZSWQZ
|
6.7 | Ki | 41 | — | |
XYLJTJTWOPEYJR
|
6.7 | Kd | 5 | — | |
ZVWRFVCNQOECJS
|
6.7 | Ki | 71 | — | |
CPHGZDSYMREPNQ
|
6.7 | IC50 | 6 | — | |
DTKNQMRYSGVPEX
|
6.7 | IC50 | 3 | — | |
IBWUYNSLISMPFY
|
6.7 | IC50 | 4 | — | |
NRQSCGVAXSQZCR
|
6.7 | IC50 | 4 | — | |
RXPZOSHFGJWSLQ
|
6.7 | IC50 | 6 | — | |
NCDRKKZNMOSYQQ
|
6.7 | IC50 | 2 | — | |
GCDSDVNITVBCDW
|
6.6 | IC50 | 17 | — | |
NXSJMRCTGYTSTK
|
6.6 | Kd | 200 | — | |
NHHQJBCNYHBUSI
|
6.6 | Kd | 220 | — | |
GRALRZJBEGFAHQ
|
6.6 | IC50 | 2 | — | |
HDRLAVNNWSHSOA
|
6.6 | Ki | 19 | — | |
RTDSHUGNRVXRHN
|
6.6 | Ki | 51 | — | |
VWACUNWBMWWMPJ
|
6.6 | Ki | 18 | — | |
XOOAAYRIVATZNM
|
6.6 | Ki | 55 | — | |
XQVVPGYIWAGRNI
|
6.6 | Ki | 19 | — | |
ZWVZORIKUNOTCS
|
6.6 | Ki | 69 | — | |
UJBJWYNPUOLFIZ
|
6.6 | IC50 | 49 | — |