Target Details
| UniProt AC | Q9UM73 |
|---|---|
| Gene Symbol | ALK |
| Protein Name | ALK tyrosine kinase receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12810 (ALK_LTK_GRD) PF00629 (MAM) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 712
- Clinical molecules 27
- Avg pChEMBL 7.64
KEGG Pathways (3)
Associated Diseases (4)
Active Molecules (712)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GXJSLIOOPZRPEV
|
7.1 | Ki | 34 | — | |
NRFMLFPXDKIQBF
|
7.1 | Kd | 8 | — | |
OBVABXWHTLZJKU
|
7.1 | IC50 | 2 | — | |
QLNWZYTUBBNBEL
|
7.1 | IC50 | 2 | — | |
WBQBMMMQJSJEJT
|
7.1 | Ki | 4 | — | |
JINIKYUAUCGQAS
|
7.1 | IC50 | 3 | — | |
OZNRQZFKHOJXCQ
|
7.1 | IC50 | 2 | — | |
JQWJRFOFKDLCQB
|
7.1 | IC50 | 2 | — | |
JZMFNCMUNMDDDE
|
7.1 | IC50 | 2 | — | |
TWABWUVZWXSPTC
|
7.1 | IC50 | 3 | — | |
VCLHKFSMXAYHRB
|
7.1 | IC50 | 2 | — | |
BNXYQBUYYXJKBW
|
7.1 | IC50 | 3 | — | |
DOWWFGLYJNBUSG
|
7.1 | IC50 | 4 | — | |
JXPQCRCHIRKWDH
|
7.1 | IC50 | 3 | — | |
NVTUEJKEIISOPJ
|
7.1 | IC50 | 3 | — | |
POXSFRWIBWNONT
|
7.1 | IC50 | 3 | — | |
RONLQWJKAFWDOO
|
7.1 | IC50 | 3 | — | |
VPYPBQZXCLHXPF
|
7.1 | IC50 | 3 | — | |
YNXUIZMRPVCJTM
|
7.1 | IC50 | 3 | — | |
SHRNMJSKKQHLKT
|
7.0 | IC50 | 4 | — | |
UWQCPRVJOPGITM
|
7.0 | IC50 | 2 | — | |
KGHHVSJZWGWWDG
|
7.0 | IC50 | 4 | Yes | |
MFBMGGILJVFTKT
|
7.0 | IC50 | 2 | — | |
UDVJBRYBBSVDDS
|
7.0 | IC50 | 14 | — | |
UMBIRSZUCJNBHB
|
7.0 | IC50 | 18 | — | |
DEIJESKINOLXTC
|
7.0 | IC50 | 2 | — | |
GIBYRJLRSLPQGP
|
7.0 | IC50 | 6 | — | |
NSKYYUZMAXEZIR
|
7.0 | Ki | 15 | — | |
QDCQSLLXPYSDTE
|
7.0 | IC50 | 2 | — | |
WHUMNDGRLJYAMI
|
7.0 | IC50 | 2 | — | |
COPINYWCESNOFK
|
7.0 | IC50 | 3 | — | |
FLEAYYMORDPWAJ
|
7.0 | Ki | 90 | — | |
NRGYZNJPCGRCLV
|
7.0 | Ki | 52 | — | |
QXIOZIFTPMAING
|
7.0 | IC50 | 17 | — | |
RGNHKJWHFIPHIM
|
7.0 | Ki | 66 | — | |
RYYNGWLOYLRZLK
|
7.0 | Ki | 104 | — | |
ZCICFBOTBSKMJF
|
7.0 | IC50 | 2 | — | |
JBRATJAZJLQBMD
|
7.0 | IC50 | 2 | — | |
OIEHQPKUMMPJDV
|
7.0 | IC50 | 2 | — | |
ANDWXAGCNLNBJR
|
7.0 | IC50 | 2 | — | |
PCIMPOMGHFNGMS
|
6.9 | IC50 | 7 | — | |
SXEYAAMYAQFZGM
|
6.9 | IC50 | 2 | — | |
JXNMCDLXYWQTIW
|
6.9 | Ki | 13 | — | |
KHGPYYFCIAISBU
|
6.9 | Ki | 31 | — | |
LBVKEEFIPBQIMD
|
6.9 | Ki | 27 | — | |
PROLIXHVRCJEFH
|
6.9 | Ki | 46 | — | |
QYFQPPSZJOXIML
|
6.9 | Ki | 3 | — | |
BMWIOANJDKPITJ
|
6.9 | IC50 | 4 | — | |
YBYZNVHZPUSHTD
|
6.9 | IC50 | 2 | — | |
LVYXERPKYAQGKM
|
6.8 | IC50 | 4 | — |