Target Details
| UniProt AC | Q9UM73 |
|---|---|
| Gene Symbol | ALK |
| Protein Name | ALK tyrosine kinase receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12810 (ALK_LTK_GRD) PF00629 (MAM) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 712
- Clinical molecules 27
- Avg pChEMBL 7.64
KEGG Pathways (3)
Associated Diseases (4)
Active Molecules (712)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UNCWKKAXUDLWHL
|
7.3 | IC50 | 2 | — | |
HYVDZBWKEAFWAG
|
7.3 | IC50 | 2 | — | |
IHCBPZKNVNJFAT
|
7.3 | IC50 | 2 | — | |
KTEIFNKAUNYNJU
|
7.3 | IC50 | 48 | — | |
PYYVZOAOTZMECL
|
7.3 | IC50 | 2 | — | |
ABKGHWKSGAOXGR
|
7.3 | IC50 | 2 | — | |
AKWLDQDWZNJYKL
|
7.3 | IC50 | 14 | — | |
DBXGGXLBTWZXBB
|
7.3 | Ki | 39 | — | |
LCGSWTFWYNYUKS
|
7.3 | Ki | 26 | — | |
MVJMMLFMPWITEJ
|
7.3 | Ki | 110 | — | |
QHXBWJSQXSYAGG
|
7.3 | IC50 | 16 | — | |
RKSKGSQDRZHVPG
|
7.3 | IC50 | 2 | — | |
VGEDWONGQUXJQA
|
7.3 | IC50 | 7 | — | |
ABDKJOVFIDLNSS
|
7.3 | IC50 | 2 | — | |
IBUOCLLDDGZTCA
|
7.3 | IC50 | 2 | — | |
HAYYBYPASCDWEQ
|
7.3 | IC50 | 47 | — | |
LIWMTOPLJLFZKX
|
7.3 | IC50 | 2 | — | |
ZLEPBLGJEZUDSL
|
7.2 | IC50 | 2 | — | |
RTQRIPALPGYRNN
|
7.2 | IC50 | 2 | — | |
FXUVMEINVSOBBC
|
7.2 | IC50 | 4 | — | |
AEKJPCHGTMQXDQ
|
7.2 | IC50 | 2 | — | |
CAHIYUNFMZWRQZ
|
7.2 | IC50 | 2 | — | |
QXAZYKBUUHKHCE
|
7.2 | IC50 | 4 | — | |
YKKMSYLSEXFJCA
|
7.2 | IC50 | 2 | — | |
GQGMUKOYILWOIQ
|
7.2 | Ki | 25 | — | |
HBJUFAHIACMPFY
|
7.2 | Ki | 4 | — | |
HZPACYSNLOCDLW
|
7.2 | Ki | 48 | — | |
IJNMRIYHRCSVCO
|
7.2 | IC50 | 3 | — | |
JZTOUVBEZONDKA
|
7.2 | Ki | 80 | — | |
LSSNCWGAWKTCBU
|
7.2 | Ki | 2 | — | |
TVUWQDLBEOZVOU
|
7.2 | Ki | 41 | — | |
VKBFHTIUXUCYRQ
|
7.2 | Ki | 66 | — | |
BUHLWVQDHMLTPT
|
7.2 | IC50 | 2 | — | |
CCASRZWPCOLUMW
|
7.2 | IC50 | 3 | — | |
PZPRNRYGJJTJJT
|
7.2 | IC50 | 2 | — | |
SHZQPUOQOSUSFR
|
7.2 | IC50 | 2 | — | |
XSJJLTUTXVNLLI
|
7.2 | IC50 | 3 | — | |
CXQHYVUVSFXTMY
|
7.2 | Kd | 154 | — | |
JZLUCFJMWJDRIK
|
7.2 | IC50 | 7 | — | |
MOWRRSWYFUOCAR
|
7.2 | IC50 | 3 | — | |
PZZSEHAIVIYFLT
|
7.2 | IC50 | 2 | — | |
SEJGTFPOEJWEGG
|
7.2 | Kd | 149 | — | |
UIARLYUEJFELEN
|
7.2 | Kd | 289 | Yes | |
MATHWQFCWXKDBA
|
7.1 | IC50 | 2 | — | |
FXGUUNXTWGWEDY
|
7.1 | IC50 | 3 | — | |
WQTDKOSNNMUDQK
|
7.1 | IC50 | 5 | — | |
LBMWDLUJEOLXOE
|
7.1 | IC50 | 2 | — | |
QSUYIPABXMWKIL
|
7.1 | IC50 | 2 | — | |
ZOUKGWPEJXISGG
|
7.1 | IC50 | 2 | — | |
AIQDZMUPVYDVLB
|
7.1 | Ki | 48 | — |