Target Details
| UniProt AC | Q9UM73 |
|---|---|
| Gene Symbol | ALK |
| Protein Name | ALK tyrosine kinase receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12810 (ALK_LTK_GRD) PF00629 (MAM) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 712
- Clinical molecules 27
- Avg pChEMBL 7.64
KEGG Pathways (3)
Associated Diseases (4)
Active Molecules (712)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OIIPLUSQGIIGMV
|
10.0 | IC50 | 2 | — | |
XBAUQTADQOFONU
|
9.9 | IC50 | 3 | — | |
CBCRRZVVZMJUTF
|
9.7 | IC50 | 3 | — | |
YHWJHUBPWLCING
|
9.7 | IC50 | 3 | — | |
RQDNRYSBNFWQCV
|
9.7 | IC50 | 3 | — | |
PLCZCZWCIOPXGS
|
9.6 | IC50 | 3 | — | |
XIQAFZIFYBEQQW
|
9.6 | IC50 | 3 | — | |
UMIDCBQSQODODG
|
9.6 | IC50 | 3 | — | |
QSLMZWGPJXKPBS
|
9.6 | IC50 | 3 | — | |
BHLTVGNUTOSHBD
|
9.5 | IC50 | 3 | — | |
HFTHUIUDNIONGS
|
9.5 | IC50 | 3 | — | |
QVMUQQQYQHYSBY
|
9.5 | IC50 | 2 | — | |
YRUIXESBPXQWOD
|
9.5 | IC50 | 3 | — | |
ZKSMNJVVPOADIE
|
9.5 | IC50 | 3 | — | |
CCVGHLZQHJYDAI
|
9.4 | IC50 | 3 | — | |
IWKVFBINMMDGNH
|
9.4 | IC50 | 3 | — | |
HBAGNJCIEGUKLI
|
9.4 | IC50 | 2 | — | |
FLTJPMCKNUNPRH
|
9.4 | IC50 | 3 | — | |
ZTKZGNHMDMISHE
|
9.4 | IC50 | 3 | — | |
SWDUUFOEGXYQAO
|
9.3 | IC50 | 3 | — | |
ZRFJCNOHKKQRSS
|
9.3 | IC50 | 3 | — | |
HXZDICYKFAOZLE
|
9.3 | IC50 | 6 | Yes | |
HZTYDQRUAWIZRE
|
9.3 | IC50 | 40 | Yes | |
KJWZHCRQZUOQJR
|
9.3 | IC50 | 3 | — | |
LZNLVKVRHVELDP
|
9.3 | IC50 | 3 | — | |
OGBBOXLWGHVVPQ
|
9.2 | IC50 | 3 | — | |
ZCTVEBRXLFXVIK
|
9.2 | IC50 | 3 | — | |
NFZBAKHCVIQLBD
|
9.2 | IC50 | 2 | — | |
XNRABRXYGRUDAX
|
9.2 | IC50 | 3 | — | |
RPUSLEYUMRGACQ
|
9.2 | IC50 | 3 | — | |
XRVFEWYOEIYZGB
|
9.2 | IC50 | 3 | — | |
ASQDMAQHZGURLM
|
9.2 | IC50 | 2 | — | |
ASQDMAQHZGURLM
|
9.2 | IC50 | 2 | — | |
FJSAYHJPHADVOT
|
9.2 | IC50 | 2 | — | |
VXYZCOCRVAQWBG
|
9.2 | Ki | 15 | — | |
MQCNUAFNUAISQK
|
9.1 | IC50 | 3 | — | |
GCYIGMXOIWJGBU
|
9.1 | Ki | 2 | — | |
WDUXPXHDIYWLHP
|
9.1 | IC50 | 3 | — | |
YUEGRPWDOBJWDW
|
9.1 | IC50 | 3 | — | |
DGIKQZFVNNRZMT
|
9.1 | IC50 | 3 | — | |
DIXMBHMNEHPFCX
|
9.1 | IC50 | 12 | — | |
LEVAPGLCIYCDDH
|
9.1 | IC50 | 3 | — | |
FXYPQFBJRKMLDS
|
9.1 | IC50 | 4 | — | |
XGZORHKVFKUMAV
|
9.1 | IC50 | 4 | — | |
KYODHQKKLBGUED
|
9.1 | IC50 | 3 | — | |
UETYAVAIGWIDEO
|
9.1 | IC50 | 3 | — | |
LFOZAGZOWUEXKO
|
9.0 | IC50 | 2 | — | |
IBXPUECEDDUZFG
|
9.0 | IC50 | 3 | — | |
GERKWUCMHZITIS
|
9.0 | IC50 | 2 | — | |
GZYCQQBRSRIFII
|
9.0 | IC50 | 7 | — |