Target Details
| UniProt AC | Q9UM47 |
|---|---|
| Gene Symbol | NOTCH3 |
| Protein Name | Neurogenic locus notch homolog protein 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF00008 (EGF) PF07645 (EGF_CA) PF12661 (hEGF) PF06816 (NOD) PF07684 (NODP) PF00066 (Notch) |
Summary
- Multi-target molecules 53
- Clinical molecules 0
- Avg pChEMBL 8.29
KEGG Pathways (9)
Associated Diseases (4)
Active Molecules (53)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DYNTZUXZTDSIOF
|
7.2 | IC50 | 2 | — | |
WGYNBTCNYOMMNG
|
6.9 | IC50 | 2 | — | |
RMRHTXFKXWUOFV
|
6.8 | IC50 | 2 | — |