Target Details
| UniProt AC | Q9ULW0 |
|---|---|
| Gene Symbol | TPX2 |
| Protein Name | Targeting protein for Xklp2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF09041 (Aurora-A_bind) PF06886 (TPX2) PF12214 (TPX2_importin) |
Summary
- Multi-target molecules 22
- Clinical molecules 13
- Avg pChEMBL 7.01
Active Molecules (22)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ULOLUGXMKLIZGE
|
8.2 | IC50 | 8 | Yes | |
QWJHWNIFEWOQTF
|
8.1 | IC50 | 5 | Yes | |
YRIZEPGWRQGUBO
|
7.8 | IC50 | 4 | Yes | |
AORICYPGAMGKBS
|
7.8 | Kd | 2 | — | |
ABQBTGKORANNEM
|
7.7 | Kd | 2 | — | |
WKDACQVEJIVHMZ
|
7.7 | IC50 | 46 | — | |
DZICJKNDYKNBTO
|
7.4 | IC50 | 4 | Yes | |
XIZHRWKYFLKHBC
|
7.2 | IC50 | 4 | Yes | |
ZCEDSBRRQLSVCI
|
7.2 | Kd | 2 | — | |
WVYZESHCWKLDBS
|
7.1 | IC50 | 5 | Yes | |
ANQYGKVLKNBYFQ
|
7.1 | Kd | 2 | — | |
KVLWDVXAVQTEGW
|
7.0 | Kd | 2 | — | |
MENIKIFJGYYVNI
|
6.9 | IC50 | 5 | Yes | |
SCRSXZZGUOEUBI
|
6.8 | IC50 | 4 | Yes | |
HXZMDXUYYVDPRW
|
6.8 | Kd | 2 | — | |
WKRMVDGCONSBRA
|
6.7 | Kd | 2 | — | |
QTBWCSQGBMPECM
|
6.3 | Ki | 21 | Yes | |
FATFDRYYCYZBQB
|
6.2 | IC50 | 5 | Yes | |
FFNIWOOLZGAOAB
|
6.2 | IC50 | 8 | Yes | |
GASPHORHXIOCBB
|
6.0 | IC50 | 4 | Yes | |
LOEVXPKFXLHBHC
|
6.0 | Kd | 2 | — | |
IMQVBCRZLIQNPG
|
6.0 | IC50 | 5 | Yes |