Target Details
| UniProt AC | Q9ULD4 |
|---|---|
| Gene Symbol | BRPF3 |
| Protein Name | Bromodomain and PHD finger-containing protein 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00439 (Bromodomain) PF10513 (EPL1) PF13831 (PHD_2) PF00855 (PWWP) PF13832 (zf-HC5HC2H_2) |
Summary
- Multi-target molecules 11
- Clinical molecules 0
- Avg pChEMBL 6.55
Active Molecules (11)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HYQBRUSSCIAOOD
|
7.6 | Kd | 6 | — | |
VZAFGXCWAWRULT
|
7.0 | Ki | 7 | — | |
XHAYAQCABOVSNX
|
6.9 | Kd | 9 | — | |
LQDXWIYREJVTTB
|
6.7 | IC50 | 4 | — | |
BMVCSXFOQPYKKC
|
6.6 | IC50 | 5 | — | |
XULQOMADHZABKB
|
6.5 | IC50 | 3 | — | |
UEMQPCYDWCSVCU
|
6.4 | Kd | 5 | — | |
YPOOJPDFTKZDEW
|
6.2 | IC50 | 3 | — | |
BTTCKSLDCMBUAH
|
6.1 | Ki | 7 | — | |
QCIJLRJBZDBVDB
|
6.0 | Kd | 5 | — | |
VXXXPCKZPJGNGK
|
6.0 | IC50 | 4 | — |