Target Details
| UniProt AC | Q9UL54 |
|---|---|
| Gene Symbol | TAOK2 |
| Protein Name | Serine/threonine-protein kinase TAO2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 27
- Clinical molecules 9
- Avg pChEMBL 6.55
KEGG Pathways (2)
Active Molecules (27)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DKZYXHCYPUVGAF
|
8.0 | Kd | 112 | — | |
HKSZLNNOFSGOKW
|
7.9 | IC50 | 408 | — | |
ODPGGGTTYSGTGO
|
7.4 | Kd | 153 | — | |
OVPNQJVDAFNBDN
|
7.3 | Kd | 44 | Yes | |
JWILUIVAYLRFIY
|
7.1 | IC50 | 14 | — | |
DGLFSNZWRYADFC
|
7.0 | IC50 | 12 | — | |
YRDHKIFCGOZTGD
|
6.9 | IC50 | 21 | — | |
YABJJWZLRMPFSI
|
6.8 | Kd | 34 | — | |
BIIVYFLTOXDAOV
|
6.6 | Kd | 82 | Yes | |
HFNKQEVNSGCOJV
|
6.5 | Kd | 65 | — | |
MFAQYJIYDMLAIM
|
6.4 | Kd | 130 | Yes | |
LYADGAGFYYXXIO
|
6.4 | IC50 | 82 | — | |
GCIKSSRWRFVXBI
|
6.4 | Kd | 109 | Yes | |
VAARYSWULJUGST
|
6.4 | Kd | 119 | Yes | |
UIARLYUEJFELEN
|
6.3 | Kd | 289 | Yes | |
UJBJWYNPUOLFIZ
|
6.3 | IC50 | 49 | — | |
MLDQJTXFUGDVEO
|
6.3 | Kd | 85 | Yes | |
NHHQJBCNYHBUSI
|
6.2 | Kd | 220 | — | |
DCYHJVFMNYSPNT
|
6.2 | IC50 | 9 | — | |
QQWUGDVOUVUTOY
|
6.1 | Kd | 231 | Yes | |
JOOXLOJCABQBSG
|
6.1 | Kd | 139 | — | |
JRNJNYBQQYBCLE
|
6.1 | Kd | 40 | Yes | |
KTEIFNKAUNYNJU
|
6.0 | Kd | 114 | — | |
WPXVVAWAHQHJPF
|
6.0 | IC50 | 41 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |