Target Details
| UniProt AC | Q9UKP4 |
|---|---|
| Gene Symbol | ADAMTS7 |
| Protein Name | A disintegrin and metalloproteinase with thrombospondin motifs 7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17771 (ADAMTS_CR_2) PF19236 (ADAMTS_CR_3) PF05986 (ADAMTS_spacer1) PF01562 (Pep_M12B_propep) PF01421 (Reprolysin) PF19030 (TSP1_ADAMTS) PF00090 (TSP_1) |
Summary
- Multi-target molecules 16
- Clinical molecules 0
- Avg pChEMBL 7.81
Active Molecules (16)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OBXOKKGDFARJJV
|
8.8 | IC50 | 2 | — | |
JPZUAZMIFKHSGZ
|
8.6 | IC50 | 2 | — | |
QOPRVQPJWCZITD
|
8.6 | IC50 | 2 | — | |
RPVHARCGZZMFFN
|
8.6 | IC50 | 2 | — | |
WNKWHJMCHLXGLE
|
8.5 | IC50 | 2 | — | |
BSYDZRAGBLIBSI
|
8.5 | IC50 | 2 | — | |
LPQXZOJIUVOCAL
|
8.2 | IC50 | 2 | — | |
ZRQWUQCXSKEXGA
|
8.2 | Ki | 6 | — | |
ITOCNBUUDLLSTD
|
7.4 | Ki | 2 | — | |
MYNRCIAHZNZKOZ
|
7.4 | Ki | 2 | — | |
DAWHPQGJJMGZKV
|
7.3 | Ki | 2 | — | |
GNBHJTYIJMLFLC
|
7.3 | IC50 | 6 | — | |
WZJSIDSSGZFOCC
|
7.3 | Ki | 2 | — | |
GYSTVJYXBPSVIF
|
7.2 | Ki | 4 | — | |
JHBAOENFEKRBLY
|
6.7 | Ki | 2 | — | |
PLZHEWIMJLHYQI
|
6.4 | Ki | 2 | — |