Target Details
| UniProt AC | Q9UKL0 |
|---|---|
| Gene Symbol | RCOR1 |
| Protein Name | REST corepressor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01448 (ELM2) PF00249 (Myb_DNA-binding) PF20878 (REST_helical) |
Summary
- Multi-target molecules 149
- Clinical molecules 0
- Avg pChEMBL 6.99
KEGG Pathways (1)
Active Molecules (149)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XAHKAVMFHXJCHB
|
6.7 | IC50 | 2 | — | |
GTROCWLWUVDATG
|
6.7 | Kd | 2 | — | |
HPOREVJOPMPYMP
|
6.7 | IC50 | 2 | — | |
QAWFHNZRRCAPTH
|
6.7 | IC50 | 2 | — | |
BGINPISVOPSPQR
|
6.7 | IC50 | 2 | — | |
QQPOJEUOIDVOMC
|
6.7 | Ki | 2 | — | |
OATSDCVSNMRNCF
|
6.6 | Kd | 2 | — | |
PIBPGIZBVJIBSO
|
6.6 | Kd | 2 | — | |
PKEMMZZQSKPHHM
|
6.6 | IC50 | 2 | — | |
SSWIQIUOBLUKHT
|
6.6 | IC50 | 3 | — | |
WERQTKVJYYYSJV
|
6.6 | IC50 | 2 | — | |
GMXYXMQFGWCTDH
|
6.6 | Kd | 2 | — | |
VJBZUQSLIWXRQB
|
6.6 | IC50 | 2 | — | |
YYFDMPHIONBOKZ
|
6.6 | Kd | 3 | — | |
BESZCCPLVFYBMF
|
6.6 | Kd | 2 | — | |
MDWIPEDOGYFSLP
|
6.6 | IC50 | 2 | — | |
WEIBITIUXRSXKV
|
6.6 | IC50 | 2 | — | |
ZNYZYOQPSXVGPS
|
6.6 | IC50 | 2 | — | |
IPBBEAIDXLVCLZ
|
6.6 | IC50 | 2 | — | |
VNXLMJGQXWEBFC
|
6.6 | IC50 | 3 | — | |
WLEYRXSEUCAWFN
|
6.5 | IC50 | 2 | — | |
CIBIPCOECWRQSS
|
6.5 | IC50 | 2 | — | |
WTBPQDAPAUFMAX
|
6.5 | IC50 | 2 | — | |
HRBNXEOQKKAVFW
|
6.5 | IC50 | 2 | — | |
NAKRWHICVCPKFI
|
6.5 | IC50 | 2 | — | |
WDWILUYBYWRTDI
|
6.5 | IC50 | 3 | — | |
TYTLARZOLKJSJU
|
6.5 | IC50 | 3 | — | |
TYTLARZOLKJSJU
|
6.5 | IC50 | 3 | — | |
BCPQOLODGAYAFW
|
6.5 | IC50 | 2 | — | |
WZCZPTMDQMQDAD
|
6.5 | IC50 | 2 | — | |
LVDVKDUVNVPLJS
|
6.5 | IC50 | 2 | — | |
DCKSUHOUTHQLSM
|
6.5 | IC50 | 2 | — | |
SSKYMUOQDBRVKO
|
6.4 | Kd | 2 | — | |
NMUJNKCEYQHYGT
|
6.4 | IC50 | 2 | — | |
LTIMUTHHZPKOSE
|
6.3 | Kd | 2 | — | |
SPGITBIVGNUZCH
|
6.3 | IC50 | 2 | — | |
WQVJHHACXVLGBL
|
6.3 | Kd | 2 | — | |
AQIQXAQNDASVRZ
|
6.3 | IC50 | 6 | — | |
GOTQEJNZEOHNAE
|
6.3 | IC50 | 2 | — | |
ISNHLBSSCQSOIX
|
6.2 | IC50 | 2 | — | |
PKPPVRKPLWFXFM
|
6.2 | Ki | 2 | — | |
PSHJCIYTQFLPRP
|
6.2 | IC50 | 2 | — | |
BAJBBYYUVNGYKO
|
6.2 | IC50 | 2 | — | |
KBPKNXJNAIWYOS
|
6.1 | IC50 | 2 | — | |
CMAZUZORDXKXGI
|
6.1 | IC50 | 2 | — | |
BDCFRHXPQHIPOB
|
6.1 | IC50 | 2 | — | |
YHLPIXATFAHNPC
|
6.1 | IC50 | 2 | — | |
ZMGVXQYQAOSCBG
|
6.0 | Kd | 2 | — | |
REOMUUQHANEINM
|
6.0 | IC50 | 2 | — |