Target Details
| UniProt AC | Q9UKL0 |
|---|---|
| Gene Symbol | RCOR1 |
| Protein Name | REST corepressor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01448 (ELM2) PF00249 (Myb_DNA-binding) PF20878 (REST_helical) |
Summary
- Multi-target molecules 149
- Clinical molecules 0
- Avg pChEMBL 6.99
KEGG Pathways (1)
Active Molecules (149)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ALHBJBCQLJZYON
|
9.2 | IC50 | 4 | — | |
NTRMVYTYDOLCRU
|
8.7 | IC50 | 2 | — | |
QZNGFWQWWSECMG
|
8.5 | IC50 | 2 | — | |
VUPIIHSYRDZCSU
|
8.4 | IC50 | 2 | — | |
CTRYUUQZYMUPNG
|
8.3 | IC50 | 2 | — | |
ALHBJBCQLJZYON
|
8.2 | IC50 | 3 | — | |
XTIUXFVWQDSKHY
|
8.2 | IC50 | 2 | — | |
ZNPKDAJYJOBTSM
|
8.1 | IC50 | 2 | — | |
ZZLBFEKJJDCLHD
|
8.1 | IC50 | 2 | — | |
SQSNNQXVJVEDMY
|
8.1 | IC50 | 2 | — | |
ZPIXRPPZFQFTJS
|
8.1 | IC50 | 2 | — | |
PYDFVFWGGDZAOA
|
8.0 | IC50 | 2 | — | |
OAZVHMYGOGQYLZ
|
7.8 | IC50 | 2 | — | |
FFYGOYSNGFPHEN
|
7.7 | IC50 | 3 | — | |
HQRYNOVKRKLADI
|
7.7 | IC50 | 2 | — | |
OAZVHMYGOGQYLZ
|
7.7 | IC50 | 2 | — | |
IQVDLEXWAPYWDT
|
7.7 | Kd | 2 | — | |
DDEBLIXHOWDGMM
|
7.6 | IC50 | 4 | — | |
JELFJCHCBUKLFJ
|
7.6 | IC50 | 2 | — | |
IKJFIPIKSOKVSV
|
7.5 | IC50 | 3 | — | |
KEXPXBUNMVXDSV
|
7.5 | IC50 | 2 | — | |
SRNUZUYKHZOGFL
|
7.5 | IC50 | 2 | — | |
YXTYPKDXCRBOFD
|
7.5 | IC50 | 3 | — | |
HLHUFXWETVNBDN
|
7.5 | IC50 | 3 | — | |
UGYBNTNFUXFKEE
|
7.5 | IC50 | 2 | — | |
WJUINCYWBXZRNH
|
7.4 | IC50 | 2 | — | |
OJCTVINEUNWRJO
|
7.4 | IC50 | 2 | — | |
AORRFKCUHQJLBK
|
7.4 | Ki | 2 | — | |
VLAPFESAHIUASX
|
7.4 | IC50 | 3 | — | |
FFYJSQJRMOFPKF
|
7.4 | IC50 | 3 | — | |
QZNGFWQWWSECMG
|
7.3 | IC50 | 2 | — | |
TVPSDFDZPXEOIQ
|
7.3 | IC50 | 2 | — | |
BUTMZXYDLXMRED
|
7.3 | Ki | 2 | — | |
SNZBTOXJQFMTHW
|
7.3 | Ki | 2 | — | |
XLZPYWFUNBTRGV
|
7.3 | IC50 | 3 | — | |
NSWDBAURHGVFRJ
|
7.3 | IC50 | 3 | — | |
KSNYGZADPGAMKR
|
7.2 | IC50 | 2 | — | |
SBZNZJNYVPWQPU
|
7.2 | Ki | 2 | — | |
FICFTOMKYYZSEL
|
7.2 | IC50 | 4 | — | |
JEZAGOJTCWQABS
|
7.2 | IC50 | 2 | — | |
VQXSHYNCIQFRBL
|
7.2 | IC50 | 3 | — | |
CRFTYPZVLZZIHU
|
7.2 | IC50 | 2 | — | |
IYOQBCSTSLISOI
|
7.2 | IC50 | 2 | — | |
RUFLTUCAFVGHGI
|
7.2 | IC50 | 2 | — | |
ZVVDKVJEGXSFFZ
|
7.2 | IC50 | 2 | — | |
PNLZPOBONAJYFY
|
7.2 | IC50 | 2 | — | |
DHKMEXBVLDKGIA
|
7.1 | IC50 | 2 | — | |
NXKYPBDDPFDALC
|
7.1 | IC50 | 3 | — | |
PSRVWCBORZIYDW
|
7.1 | Ki | 2 | — | |
RZPJSFNGGGHGEC
|
7.1 | IC50 | 2 | — |