Target Details
| UniProt AC | Q9UKK3 |
|---|---|
| Gene Symbol | PARP4 |
| Protein Name | Protein mono-ADP-ribosyltransferase PARP4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00533 (BRCT) PF00644 (PARP) PF26156 (PARP4_MVP-ID) PF08487 (VIT) PF00092 (VWA) PF26166 (WGR-like_PARP4) |
Summary
- Multi-target molecules 11
- Clinical molecules 0
- Avg pChEMBL 6.86
KEGG Pathways (2)
Active Molecules (11)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HWGQMRYQVZSGDQ
|
9.2 | Kd | 7 | — | |
STSCRAGBCYODMY
|
9.0 | IC50 | 8 | — | |
JNAHVYVRKWKWKQ
|
7.0 | Kd | 4 | — | |
HWGQMRYQVZSGDQ
|
6.6 | IC50 | 6 | — | |
FDLYAMZZIXQODN
|
6.4 | IC50 | 11 | — | |
AOLFJVDCFAXDOZ
|
6.4 | IC50 | 4 | — | |
PCHKPVIQAHNQLW
|
6.3 | IC50 | 8 | — | |
JNLILESBBKKTIC
|
6.3 | IC50 | 2 | — | |
GFHLWWHOLUWZLZ
|
6.2 | IC50 | 4 | — | |
UYJZZVDLGDDTCL
|
6.1 | IC50 | 8 | — | |
HMABYWSNWIZPAG
|
6.1 | IC50 | 12 | — |