Target Details
| UniProt AC | Q9UKI8 |
|---|---|
| Gene Symbol | TLK1 |
| Protein Name | Serine/threonine-protein kinase tousled-like 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 12
- Clinical molecules 3
- Avg pChEMBL 6.46
Active Molecules (12)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
7.6 | IC50 | 408 | — | |
HKSZLNNOFSGOKW
|
7.6 | Kd | 213 | — | |
UIARLYUEJFELEN
|
7.0 | Kd | 289 | Yes | |
NHHQJBCNYHBUSI
|
6.3 | Kd | 220 | — | |
AXRCEOKUDYDWLF
|
6.3 | Kd | 31 | — | |
UBPYILGKFZZVDX
|
6.2 | Kd | 130 | Yes | |
CTNPALGJUAXMMC
|
6.2 | Kd | 2 | — | |
CTNPALGJUAXMMC
|
6.2 | Kd | 151 | — | |
WINHZLLDWRZWRT
|
6.1 | Kd | 201 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |