Target Details
| UniProt AC | Q9UKE5 |
|---|---|
| Gene Symbol | TNIK |
| Protein Name | TRAF2 and NCK-interacting protein kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 163
- Clinical molecules 21
- Avg pChEMBL 7.23
Associated Diseases (1)
Active Molecules (163)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FCHBYZITXHHPQO
|
6.3 | IC50 | 2 | — | |
KRIUNPBAQZGFQA
|
6.3 | Kd | 76 | — | |
PGFXFAOPCBAZDE
|
6.3 | IC50 | 2 | — | |
WOSKHXYHFSIKNG
|
6.2 | Kd | 24 | — | |
ZFXGOGALEGXWEL
|
6.2 | IC50 | 5 | — | |
RYYNGWLOYLRZLK
|
6.1 | Kd | 45 | — | |
LOLPPWBBNUVNQZ
|
6.1 | Kd | 97 | Yes | |
CDMGBJANTYXAIV
|
6.1 | Kd | 34 | Yes | |
XXJWYDDUDKYVKI
|
6.1 | Kd | 52 | — | |
CVWXJKQAOSCOAB
|
6.0 | Kd | 35 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |