Target Details
| UniProt AC | Q9UKE5 |
|---|---|
| Gene Symbol | TNIK |
| Protein Name | TRAF2 and NCK-interacting protein kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 163
- Clinical molecules 21
- Avg pChEMBL 7.23
Associated Diseases (1)
Active Molecules (163)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PEOZMOGNFLONKU
|
7.0 | IC50 | 2 | — | |
ZBZMGSOMPAZJPI
|
7.0 | IC50 | 2 | — | |
UQRYTVHMQZXXFL
|
7.0 | IC50 | 2 | — | |
DYNHJHQFHQTFTP
|
7.0 | Kd | 38 | — | |
YXTUXFBKHGBPPN
|
7.0 | IC50 | 2 | — | |
IJMQBOIQHQRHNW
|
7.0 | IC50 | 2 | — | |
OOSMLYPLUCBANZ
|
6.9 | IC50 | 2 | — | |
NXSJMRCTGYTSTK
|
6.9 | Kd | 200 | — | |
TYAULGBIFWWQFM
|
6.9 | IC50 | 2 | — | |
XVUSMHCLFMFBQR
|
6.9 | IC50 | 3 | — | |
SNCZIVUNTWOQAF
|
6.9 | IC50 | 4 | — | |
CPSFZCLACXEMLI
|
6.9 | IC50 | 2 | — | |
HAMDXXRICGFPSH
|
6.9 | IC50 | 2 | — | |
NPOADWCORNFOPY
|
6.9 | IC50 | 2 | — | |
VFKKCGQRHLPCSX
|
6.9 | IC50 | 2 | — | |
BPNUQXPIQBZCMR
|
6.8 | Kd | 83 | Yes | |
JWNPDZNEKVCWMY
|
6.8 | Kd | 57 | Yes | |
MVCOAUNKQVWQHZ
|
6.8 | Kd | 54 | Yes | |
GUBJNPWVIUFSTR
|
6.8 | Kd | 103 | — | |
LAYIDHXFJBAVAV
|
6.8 | IC50 | 2 | — | |
NLNNYHCSSJWXLH
|
6.8 | IC50 | 2 | — | |
WGDZJXGKHCWRMM
|
6.8 | IC50 | 2 | — | |
YCYMKWLYOBLWHH
|
6.8 | IC50 | 2 | — | |
CLODUYRNZMIONW
|
6.8 | IC50 | 3 | — | |
JTSLALYXYSRPGW
|
6.8 | Kd | 8 | — | |
WCWUXEGQKLTGDX
|
6.8 | Kd | 22 | Yes | |
CNIKPKHTIIFUOY
|
6.8 | IC50 | 2 | — | |
OWRPRNROGDZURV
|
6.8 | IC50 | 2 | — | |
WVUNYSQLFKLYNI
|
6.8 | Kd | 46 | Yes | |
YLDDOLAWPICWDH
|
6.8 | IC50 | 2 | — | |
ALKJNCZNEOTEMP
|
6.7 | Kd | 55 | — | |
KVBPVRRXTIJVIK
|
6.7 | IC50 | 2 | — | |
RITAVMQDGBJQJZ
|
6.7 | Kd | 43 | — | |
JQLFNUDNPNFXQP
|
6.7 | IC50 | 2 | — | |
VHADCIRDAFWKDN
|
6.7 | IC50 | 2 | — | |
CXQHYVUVSFXTMY
|
6.7 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.7 | Kd | 149 | — | |
WPXVVAWAHQHJPF
|
6.7 | IC50 | 41 | — | |
XFFPRUSTZBJTSC
|
6.6 | IC50 | 2 | — | |
KELYOKFNTWCOKP
|
6.6 | IC50 | 2 | — | |
YFNWWNRZJGMDBR
|
6.6 | Kd | 35 | — | |
MFAQYJIYDMLAIM
|
6.6 | Kd | 130 | Yes | |
BBBSTZKWEGVBNW
|
6.6 | IC50 | 2 | — | |
CUIHSIWYWATEQL
|
6.5 | Kd | 61 | Yes | |
OYONTEXKYJZFHA
|
6.5 | Kd | 69 | Yes | |
BPHRYFYZZXLBST
|
6.5 | IC50 | 2 | — | |
KOONCLIJVVMZCL
|
6.5 | IC50 | 2 | — | |
ZECOHPFWGOCWLO
|
6.4 | IC50 | 5 | — | |
PHXJVRSECIGDHY
|
6.4 | Kd | 59 | — | |
VAARYSWULJUGST
|
6.4 | Kd | 119 | Yes |