Target Details
| UniProt AC | Q9UKE5 |
|---|---|
| Gene Symbol | TNIK |
| Protein Name | TRAF2 and NCK-interacting protein kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 163
- Clinical molecules 21
- Avg pChEMBL 7.23
Associated Diseases (1)
Active Molecules (163)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UBPYILGKFZZVDX
|
7.5 | Kd | 130 | Yes | |
JCOMWFYBHHOUGK
|
7.4 | IC50 | 2 | — | |
HSXHOPFVRFPEGS
|
7.4 | IC50 | 2 | — | |
MGTQMPVMKHKJAF
|
7.4 | IC50 | 2 | — | |
CJNRNQUPGPBLID
|
7.4 | IC50 | 2 | — | |
OAVGBZOFDPFGPJ
|
7.4 | Kd | 42 | Yes | |
UBPYMWXTLXKKBW
|
7.4 | IC50 | 2 | — | |
AMTPPKYFTXUVJY
|
7.4 | IC50 | 2 | — | |
RIWTUJFFSTVYPW
|
7.4 | IC50 | 6 | — | |
AIYREGHPXFOWSK
|
7.4 | IC50 | 2 | — | |
SENWNDLDAHBDSA
|
7.4 | IC50 | 2 | — | |
WWFSKAMRQLRLTJ
|
7.4 | IC50 | 2 | — | |
AVEXLWXITHDXGJ
|
7.3 | IC50 | 2 | — | |
KNAKHJWNZMAMAO
|
7.3 | IC50 | 2 | — | |
VKQYTMVZQKCCID
|
7.3 | IC50 | 2 | — | |
WCCMSFLKQHUQAF
|
7.3 | IC50 | 2 | — | |
XZXHXSATPCNXJR
|
7.3 | Kd | 165 | Yes | |
ROBNMKKERIMYQP
|
7.3 | IC50 | 2 | — | |
VHBIVOIWMNXHQR
|
7.3 | IC50 | 2 | — | |
VOYZWDQJVPQGCO
|
7.2 | IC50 | 9 | — | |
BIFCETOSTFEUQU
|
7.2 | IC50 | 2 | — | |
YJVZYDNNGQCFEQ
|
7.2 | IC50 | 2 | — | |
FTBRALICGUIRHO
|
7.2 | IC50 | 2 | — | |
PAZJYAQBBSYLRQ
|
7.2 | IC50 | 2 | — | |
VHADCIRDAFWKDN
|
7.2 | IC50 | 2 | — | |
MWTNEWVBVSRDNA
|
7.2 | IC50 | 2 | — | |
YFZOGSFWULXJTA
|
7.2 | IC50 | 2 | — | |
GOYOZLWEHBWSHT
|
7.2 | IC50 | 2 | — | |
CXMURJVCMJRHAM
|
7.2 | IC50 | 2 | — | |
WNEVOMUAXQPYDE
|
7.2 | IC50 | 2 | — | |
MSWOWUREQODTRO
|
7.2 | IC50 | 11 | — | |
ODPGGGTTYSGTGO
|
7.2 | Kd | 153 | — | |
XFEKSSMJINNJSX
|
7.2 | IC50 | 3 | — | |
AJSYWVVZBHGYEW
|
7.1 | IC50 | 2 | — | |
MWKSRKSEWLRPBL
|
7.1 | Kd | 1075 | — | |
UADCTKCTCBTSLU
|
7.1 | IC50 | 2 | — | |
IBWURMUNPBVKLR
|
7.1 | IC50 | 2 | — | |
YUVLZPSSXDFUHH
|
7.1 | IC50 | 3 | — | |
VLPQFOXQPCFHRL
|
7.1 | IC50 | 2 | — | |
CZWJLLBPWLUINU
|
7.1 | IC50 | 10 | — | |
CTNPALGJUAXMMC
|
7.0 | Kd | 151 | — | |
HWXVIOGONBBTBY
|
7.0 | Kd | 27 | — | |
RBCWFGWXMPYQSB
|
7.0 | IC50 | 2 | — | |
KXYYTXVXVOWNIG
|
7.0 | IC50 | 2 | — | |
IAYGCINLNONXHY
|
7.0 | Kd | 50 | — | |
KSOOWLORAVQWKJ
|
7.0 | IC50 | 2 | — | |
NAIUXUTZYFPOIK
|
7.0 | IC50 | 2 | — | |
RKBYYWVZFBATHQ
|
7.0 | IC50 | 12 | — | |
OSVUGUHRKMMBSE
|
7.0 | Kd | 170 | — | |
LQYGLUICAZYCHN
|
7.0 | IC50 | 2 | — |