Target Details
| UniProt AC | Q9UKE5 |
|---|---|
| Gene Symbol | TNIK |
| Protein Name | TRAF2 and NCK-interacting protein kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 163
- Clinical molecules 21
- Avg pChEMBL 7.23
Associated Diseases (1)
Active Molecules (163)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RWJSBHSWVMKBER
|
9.4 | IC50 | 2 | — | |
IAUZTOZLTFSMIE
|
9.2 | IC50 | 4 | Yes | |
ZGCQRUODVWMXSM
|
8.7 | IC50 | 2 | — | |
SRBGKBONVVVORP
|
8.6 | IC50 | 2 | — | |
VVUATAXJOVGUSR
|
8.5 | IC50 | 2 | — | |
MHEOXLMQZIYGDG
|
8.4 | IC50 | 2 | — | |
BPSYQQWLXMMBAX
|
8.4 | IC50 | 2 | — | |
FJICSOOOGVNUCL
|
8.4 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
8.3 | IC50 | 408 | — | |
HKSZLNNOFSGOKW
|
8.3 | Kd | 213 | — | |
VFLPOFHPMNYCOH
|
8.3 | IC50 | 7 | — | |
KDJJXBPORVAUEF
|
8.3 | IC50 | 2 | — | |
QKKIWEILHCXECO
|
8.3 | IC50 | 24 | — | |
UIARLYUEJFELEN
|
8.3 | Kd | 289 | Yes | |
HYUGTGGDEAGXJP
|
8.2 | IC50 | 11 | — | |
QJWIVNXPZLGILT
|
8.2 | IC50 | 2 | — | |
WTYJCTRCRZLZFE
|
8.2 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
8.1 | IC50 | 49 | Yes | |
OUCUNVKXSOPBBS
|
8.1 | IC50 | 4 | — | |
JXEPUZVUZPLZMS
|
8.0 | IC50 | 2 | — | |
KARJFNUGCLEZKM
|
8.0 | IC50 | 3 | — | |
KOZFSFOOLUUIGY
|
8.0 | Kd | 88 | Yes | |
QABFDCSQZQSQOW
|
8.0 | IC50 | 2 | — | |
ISSFPHPDMLUKPK
|
8.0 | IC50 | 2 | — | |
SIABUCJHEMLWDM
|
8.0 | IC50 | 2 | — | |
GYOQXOATKFOYNW
|
7.9 | IC50 | 2 | — | |
NHFDRBXTEDBWCZ
|
7.9 | Kd | 12 | Yes | |
RJZAPAMXDXCITJ
|
7.9 | IC50 | 2 | — | |
APXIUBHZWNOTAS
|
7.8 | IC50 | 2 | — | |
HNWRRPTZWUVJAX
|
7.8 | IC50 | 2 | — | |
KHPCIHZXOGHCLY
|
7.8 | IC50 | 3 | — | |
VBQRUKZVDRXMBF
|
7.8 | IC50 | 2 | — | |
WWWPDUVJHFVGOK
|
7.7 | IC50 | 2 | — | |
LXGDXFKSYPYLSD
|
7.7 | IC50 | 2 | — | |
QACLFFVLWCKNEA
|
7.7 | IC50 | 2 | — | |
CEOYEZFCROSXBX
|
7.6 | IC50 | 2 | — | |
NETVGXQSFUMKOX
|
7.6 | IC50 | 2 | — | |
PIQCTGMSNWUMAF
|
7.6 | Kd | 137 | Yes | |
GOUXACDXZWAKJI
|
7.6 | IC50 | 2 | — | |
TZMCWEXCNHTWOP
|
7.6 | IC50 | 2 | — | |
WINHZLLDWRZWRT
|
7.6 | Kd | 201 | Yes | |
IORLJCFZTVIEHA
|
7.6 | IC50 | 2 | — | |
RUHNYDZQGMWRMX
|
7.6 | IC50 | 2 | — | |
UVLOISNMRLZTPF
|
7.6 | IC50 | 5 | — | |
XBTZKVHEBBNOCK
|
7.6 | IC50 | 2 | — | |
ACHHYBWZGKASQH
|
7.6 | IC50 | 2 | — | |
VEMZDHGGFCZOTO
|
7.6 | IC50 | 2 | — | |
YYLKKYCXAOBSRM
|
7.5 | Kd | 191 | — | |
JHZZTEODBVPOGC
|
7.5 | IC50 | 2 | — | |
RBPNVVLVIGSUDX
|
7.5 | IC50 | 2 | — |