Target Details
| UniProt AC | Q9UK32 |
|---|---|
| Gene Symbol | RPS6KA6 |
| Protein Name | Ribosomal protein S6 kinase alpha-6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 53
- Clinical molecules 10
- Avg pChEMBL 7.03
KEGG Pathways (10)
Active Molecules (53)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.8 | IC50 | 408 | — | |
AYCPARAPKDAOEN
|
8.4 | Kd | 73 | — | |
FYXRSVDHGLUMHB
|
8.2 | IC50 | 8 | — | |
CLYZLUAUBTXCPL
|
8.2 | IC50 | 7 | — | |
MHGPJIHGGLSWFD
|
8.1 | IC50 | 8 | — | |
DWRUMXZDNGCUDK
|
8.1 | IC50 | 3 | — | |
XYMNFMNOEWBPNB
|
8.1 | IC50 | 4 | — | |
IEQAHFTVGLZUBI
|
8.0 | IC50 | 8 | — | |
IIRWNGPLJQXWFJ
|
7.9 | IC50 | 21 | — | |
OSVUGUHRKMMBSE
|
7.8 | Kd | 170 | — | |
DTEKTGDVSARYDS
|
7.8 | IC50 | 11 | — | |
LOLPPWBBNUVNQZ
|
7.8 | Kd | 97 | Yes | |
LAJAFFLJAJMYLK
|
7.7 | IC50 | 17 | — | |
NXSJMRCTGYTSTK
|
7.7 | Kd | 200 | — | |
AXRCEOKUDYDWLF
|
7.6 | Kd | 31 | — | |
RSFBRAHCHZGZPB
|
7.5 | IC50 | 8 | — | |
OZFFKOSQNBBYCA
|
7.4 | IC50 | 12 | — | |
YVQOYBIBWBAHKH
|
7.4 | IC50 | 12 | — | |
AILRADAXUVEEIR
|
7.4 | IC50 | 75 | — | |
DKZYXHCYPUVGAF
|
7.2 | Kd | 112 | — | |
QQWUGDVOUVUTOY
|
7.2 | Kd | 231 | Yes | |
YOBIWCLAYQWPPW
|
7.2 | IC50 | 23 | — | |
HIUHVDROHDSKTC
|
7.0 | Ki | 20 | — | |
UIARLYUEJFELEN
|
7.0 | Kd | 289 | Yes | |
PBCZSGKMGDDXIJ
|
6.8 | Kd | 68 | Yes | |
HFNKQEVNSGCOJV
|
6.8 | Kd | 65 | — | |
HGCJKDOLUCMPFE
|
6.8 | IC50 | 5 | — | |
XJXPKTHMXWGQPH
|
6.8 | IC50 | 5 | — | |
MZHPEELZCYWEHG
|
6.7 | IC50 | 6 | — | |
XZXHXSATPCNXJR
|
6.6 | Kd | 165 | Yes | |
UHTHHESEBZOYNR
|
6.6 | Kd | 66 | Yes | |
CDMGBJANTYXAIV
|
6.6 | Kd | 34 | Yes | |
QHKYPYXTTXKZST
|
6.6 | Kd | 28 | — | |
HZRJHVDNTDBTOZ
|
6.6 | IC50 | 8 | — | |
ZCBUQCWBWNUWSU
|
6.6 | Kd | 59 | — | |
RYYNGWLOYLRZLK
|
6.5 | Kd | 45 | — | |
ZCCPLJOKGAACRT
|
6.5 | Kd | 599 | — | |
CCQLYJZEWHWASR
|
6.5 | IC50 | 5 | — | |
ZHJGWYRLJUCMRT
|
6.5 | Kd | 18 | — | |
JOOXLOJCABQBSG
|
6.4 | Kd | 139 | — | |
BMGQWWVMWDBQGC
|
6.4 | Kd | 147 | Yes | |
BTIIUKSFWMYFNV
|
6.4 | IC50 | 6 | — | |
YYLKKYCXAOBSRM
|
6.4 | Kd | 191 | — | |
SNJRVUBJSCKVLN
|
6.3 | IC50 | 5 | — | |
UJLAWZDWDVHWOW
|
6.3 | Kd | 16 | — | |
MFAQYJIYDMLAIM
|
6.2 | Kd | 130 | Yes | |
BIIVYFLTOXDAOV
|
6.1 | Kd | 82 | Yes | |
PROGKLMIRQVLRO
|
6.1 | IC50 | 12 | — | |
WKDACQVEJIVHMZ
|
6.0 | Kd | 46 | — | |
UJIAQDJKSXQLIT
|
6.0 | Kd | 38 | — |