Target Details
| UniProt AC | Q9UIQ6 |
|---|---|
| Gene Symbol | LNPEP |
| Protein Name | Leucyl-cystinyl aminopeptidase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11838 (ERAP1_C) PF01433 (Peptidase_M1) PF17900 (Peptidase_M1_N) |
Summary
- Multi-target molecules 34
- Clinical molecules 0
- Avg pChEMBL 7.41
KEGG Pathways (1)
Active Molecules (34)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QUJXIMWUJGTUEG
|
8.7 | Ki | 2 | — | |
QCPJTEUURKCRNT
|
8.7 | IC50 | 4 | — | |
JEQPENJEYBAHIE
|
8.4 | IC50 | 3 | — | |
GSWUIYHGTPVQDP
|
8.1 | IC50 | 3 | — | |
QJVIFKMCLOJOGV
|
8.0 | IC50 | 3 | — | |
VZYRMNZEFCZSER
|
8.0 | Ki | 2 | — | |
PAISIGRMLVYIDB
|
7.9 | IC50 | 3 | — | |
WVARWRXWGWJNRJ
|
7.9 | IC50 | 3 | — | |
NJCHEVDWMWFDNQ
|
7.8 | IC50 | 3 | — | |
KFHOCODEDHRRMQ
|
7.8 | IC50 | 2 | — | |
YNFZCLOZANIMIN
|
7.7 | IC50 | 3 | — | |
WWZWLDVQUBJSGD
|
7.7 | IC50 | 3 | — | |
KAKJFMITKIMUAY
|
7.7 | IC50 | 2 | — | |
FDAGDZVCWKCEEX
|
7.6 | IC50 | 2 | — | |
FJPCLEAXXQFJFD
|
7.6 | Ki | 2 | — | |
BRDHXPSHOMSVLE
|
7.6 | Ki | 2 | — | |
SAZVKYFGANAWRA
|
7.5 | IC50 | 3 | — | |
AATVMVZMTDKRJI
|
7.5 | IC50 | 3 | — | |
ASBAZJSDHGVMRZ
|
7.5 | IC50 | 3 | — | |
BUDSAEMPVYFKML
|
7.4 | IC50 | 3 | — | |
IEYYHWFOJFXPGP
|
7.4 | IC50 | 3 | — | |
QKFOTLXPIIESQI
|
7.4 | IC50 | 5 | — | |
BUSBNAUESVLLQC
|
7.3 | IC50 | 3 | — | |
QSBGWDDCOJYQGY
|
7.2 | Ki | 4 | — | |
CDLJXXKSZOGIPE
|
7.0 | Ki | 3 | — | |
AZIAPQRBCIAHTO
|
7.0 | IC50 | 2 | — | |
HNWIOZGMMTUVKP
|
7.0 | IC50 | 2 | — | |
BUDSAEMPVYFKML
|
6.7 | IC50 | 2 | — | |
MWKSRKSEWLRPBL
|
6.5 | Kd | 1075 | — | |
WWNSEAAJQAYPMS
|
6.4 | IC50 | 2 | — | |
LCOBAHRSJLHENC
|
6.4 | IC50 | 2 | — | |
YNFZCLOZANIMIN
|
6.4 | IC50 | 2 | — | |
APTWADNFJQRAKY
|
6.2 | IC50 | 2 | — | |
JECKMXQKZJERLG
|
6.0 | IC50 | 2 | — |