Target Details
| UniProt AC | Q9UIK4 |
|---|---|
| Gene Symbol | DAPK2 |
| Protein Name | Death-associated protein kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 27
- Clinical molecules 6
- Avg pChEMBL 6.75
KEGG Pathways (3)
Active Molecules (27)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
8.8 | Kd | 213 | — | |
HKSZLNNOFSGOKW
|
8.5 | Kd | 408 | — | |
LOONVQWRKJLEEG
|
7.7 | IC50 | 8 | — | |
JOOXLOJCABQBSG
|
7.5 | Kd | 139 | — | |
NXSJMRCTGYTSTK
|
7.5 | Kd | 200 | — | |
OSVUGUHRKMMBSE
|
7.2 | Kd | 170 | — | |
NHHQJBCNYHBUSI
|
7.2 | Kd | 220 | — | |
UIARLYUEJFELEN
|
7.2 | Kd | 289 | Yes | |
NASYEGAVCTZSDO
|
7.1 | Kd | 5 | — | |
MFAQYJIYDMLAIM
|
7.0 | Kd | 130 | Yes | |
HFNKQEVNSGCOJV
|
7.0 | Kd | 65 | — | |
WINHZLLDWRZWRT
|
6.8 | Kd | 201 | Yes | |
YQMFNWQNASFQAE
|
6.8 | IC50 | 5 | — | |
CTNPALGJUAXMMC
|
6.4 | Kd | 151 | — | |
ZJQWORQRPDYKRS
|
6.3 | Kd | 7 | — | |
LIMMMAWLSIHXGX
|
6.2 | IC50 | 5 | — | |
VVFCWFGNLTVHBL
|
6.2 | IC50 | 5 | — | |
XKQNBVAZAFAZFL
|
6.2 | IC50 | 6 | — | |
KRIUNPBAQZGFQA
|
6.2 | Kd | 76 | — | |
QVJYGMLAIWRCFT
|
6.1 | IC50 | 5 | — | |
QQWUGDVOUVUTOY
|
6.1 | Kd | 231 | Yes | |
BMGQWWVMWDBQGC
|
6.0 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.0 | Kd | 91 | Yes | |
XQVVPGYIWAGRNI
|
6.0 | Kd | 34 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |