Target Details
| UniProt AC | Q9UHI8 |
|---|---|
| Gene Symbol | ADAMTS1 |
| Protein Name | A disintegrin and metalloproteinase with thrombospondin motifs 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17771 (ADAMTS_CR_2) PF19236 (ADAMTS_CR_3) PF05986 (ADAMTS_spacer1) PF01562 (Pep_M12B_propep) PF01421 (Reprolysin) PF19030 (TSP1_ADAMTS) PF00090 (TSP_1) |
Summary
- Multi-target molecules 6
- Clinical molecules 2
- Avg pChEMBL 6.76
Active Molecules (6)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZRQWUQCXSKEXGA
|
7.5 | Ki | 6 | — | |
GNBHJTYIJMLFLC
|
7.2 | Ki | 6 | — | |
LTVIJEFEZVFIST
|
7.1 | IC50 | 14 | Yes | |
SZEOXTMGYZKQHV
|
6.5 | IC50 | 4 | — | |
PWTMEJOXAUSTDY
|
6.2 | IC50 | 4 | — | |
BODLESUVCQEUII
|
6.1 | Ki | 7 | Yes |