Target Details
| UniProt AC | Q9UHD2 |
|---|---|
| Gene Symbol | TBK1 |
| Protein Name | Serine/threonine-protein kinase TBK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18394 (TBK1_CCD1) PF18396 (TBK1_ULD) |
Summary
- Multi-target molecules 639
- Clinical molecules 19
- Avg pChEMBL 7.59
KEGG Pathways (25)
- Alcoholic liver disease
- Amyotrophic lateral sclerosis
- Autophagy - animal
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Pathways of neurodegeneration - multiple diseases
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Shigellosis
- Toll-like receptor signaling pathway
- Yersinia infection
Associated Diseases (3)
Active Molecules (639)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NLHGPDUHURNAHF
|
7.2 | IC50 | 3 | — | |
XHGRACBJXGTCJY
|
7.2 | IC50 | 2 | — | |
ILQIMLNGGBJZNP
|
7.2 | IC50 | 2 | — | |
JOPQBRQUFRAGQH
|
7.2 | IC50 | 2 | — | |
XEHKYAPSLVQNOG
|
7.2 | IC50 | 2 | — | |
RDROKTFULACVDQ
|
7.2 | IC50 | 8 | — | |
OOZSAGRBHKWOLQ
|
7.2 | IC50 | 2 | — | |
VOYZWDQJVPQGCO
|
7.2 | IC50 | 9 | — | |
CFBXWHPXNROFFK
|
7.2 | IC50 | 4 | — | |
HYKUTXSZGOOHPE
|
7.2 | IC50 | 2 | — | |
LXKLPOKJWLBIKC
|
7.2 | IC50 | 2 | — | |
PECFUAQQLXEZJY
|
7.2 | IC50 | 2 | — | |
FOTACNUKABBYFV
|
7.2 | IC50 | 3 | Yes | |
VSJOESPDNYTXFI
|
7.2 | IC50 | 2 | — | |
DUBHPLWTLUVGNU
|
7.1 | IC50 | 5 | — | |
IFIYTVUHPORWKB
|
7.1 | IC50 | 3 | — | |
UDQFLASTRAMKLW
|
7.1 | IC50 | 3 | — | |
KGMZRZBOGQECSK
|
7.1 | IC50 | 2 | — | |
RYYNGWLOYLRZLK
|
7.1 | Kd | 45 | — | |
BWKLZGQQSYIAEL
|
7.1 | IC50 | 2 | — | |
KNVOICXEDILAGT
|
7.1 | Ki | 17 | — | |
PROLIXHVRCJEFH
|
7.1 | Ki | 46 | — | |
DGPQTKIPTWLNAJ
|
7.1 | IC50 | 2 | — | |
LDTAHRLHGHFHKP
|
7.1 | IC50 | 3 | — | |
XXSJUYSLBGBRGF
|
7.1 | IC50 | 2 | — | |
BXMGOFSMDOETKZ
|
7.1 | IC50 | 2 | — | |
OUTINXWZDNJANR
|
7.1 | IC50 | 2 | — | |
UOFZOMWGIVJIKW
|
7.1 | IC50 | 3 | — | |
ASDFEOAEPCPHHU
|
7.0 | IC50 | 2 | — | |
KLUCDSGOLCBPFE
|
7.0 | IC50 | 3 | — | |
QSNAYNYUEDJOLU
|
7.0 | IC50 | 2 | — | |
JOOXLOJCABQBSG
|
7.0 | Kd | 139 | — | |
SSAUMSLDIATKRC
|
7.0 | IC50 | 3 | — | |
ULGOPTXVFIQHMI
|
7.0 | IC50 | 3 | — | |
BYGZCGOGQACGKA
|
7.0 | IC50 | 2 | — | |
GUJCSPVLKMVZMJ
|
7.0 | IC50 | 3 | — | |
YOUNKSLLTJRACV
|
7.0 | IC50 | 2 | — | |
OGCZIWWQVLKYDK
|
7.0 | IC50 | 2 | — | |
UYIHWPCEDZKSLA
|
7.0 | IC50 | 2 | — | |
WNLZXWKRUIEXHK
|
7.0 | IC50 | 2 | — | |
DGEFLIVVPLYQKC
|
7.0 | IC50 | 2 | — | |
LIYOMPYVPWOZJX
|
7.0 | IC50 | 2 | — | |
UDLCUPNAFTWKLG
|
7.0 | IC50 | 2 | — | |
XMFSUNMVGUQZBX
|
7.0 | IC50 | 2 | — | |
FQMLNDAGKXRMPL
|
7.0 | IC50 | 2 | — | |
LOLPPWBBNUVNQZ
|
7.0 | Kd | 97 | Yes | |
BRHAIUXYHUZNFP
|
7.0 | IC50 | 2 | — | |
SYMILEXMAHCATG
|
7.0 | IC50 | 4 | — | |
GRIONNZJVZNNLU
|
7.0 | IC50 | 2 | — | |
NDSBUHYDEKJESH
|
7.0 | IC50 | 2 | — |