Target Details
| UniProt AC | Q9UHD2 |
|---|---|
| Gene Symbol | TBK1 |
| Protein Name | Serine/threonine-protein kinase TBK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18394 (TBK1_CCD1) PF18396 (TBK1_ULD) |
Summary
- Multi-target molecules 639
- Clinical molecules 19
- Avg pChEMBL 7.59
KEGG Pathways (25)
- Alcoholic liver disease
- Amyotrophic lateral sclerosis
- Autophagy - animal
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Pathways of neurodegeneration - multiple diseases
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Shigellosis
- Toll-like receptor signaling pathway
- Yersinia infection
Associated Diseases (3)
Active Molecules (639)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WSZQEIWUWGBMDJ
|
7.5 | IC50 | 2 | — | |
LARUOSVANYWRFG
|
7.5 | IC50 | 2 | — | |
LQABZRGBAHLOEB
|
7.5 | IC50 | 2 | — | |
QCTBKGPTHUVEKR
|
7.5 | IC50 | 2 | — | |
QKAVQJBBCRMGMX
|
7.5 | IC50 | 3 | — | |
CGFPGAHHLFCHCL
|
7.5 | IC50 | 2 | — | |
NTPUVYZJBMHFDY
|
7.5 | IC50 | 2 | — | |
OVAKBHHHFBDHMH
|
7.5 | IC50 | 2 | — | |
UKBGBACORPRCGG
|
7.5 | Kd | 17 | — | |
AWDVCHUEOUFQEL
|
7.5 | IC50 | 2 | — | |
BWUXLVAYVBIOEY
|
7.5 | IC50 | 2 | — | |
SYMILEXMAHCATG
|
7.5 | IC50 | 2 | — | |
MUOKSQABCJCOPU
|
7.5 | IC50 | 36 | — | |
YPWCKOYUDFFQRI
|
7.5 | IC50 | 2 | — | |
LLHGFGUOUWJTLQ
|
7.4 | IC50 | 3 | — | |
VFLKTHYBJXRFGI
|
7.4 | IC50 | 3 | — | |
GANHRJNVDOQXBZ
|
7.4 | IC50 | 2 | — | |
VJMPKACKJOXZGT
|
7.4 | IC50 | 2 | — | |
LPISIKGCJPHMTC
|
7.4 | IC50 | 2 | — | |
RYGAYBGVUQJRJA
|
7.4 | IC50 | 3 | — | |
XVLUNMSWJVTNRP
|
7.4 | IC50 | 4 | — | |
OWRXHGAFWZFFCW
|
7.4 | Ki | 113 | — | |
RWFVTYXPQZEJCN
|
7.4 | IC50 | 3 | — | |
FOXLRMNNJOHKBL
|
7.4 | IC50 | 2 | — | |
VCINJUXSDKRSQQ
|
7.4 | IC50 | 2 | — | |
HWCQSDRAAGDSRX
|
7.4 | IC50 | 2 | — | |
FXKNBVDEHBSMEE
|
7.4 | IC50 | 2 | — | |
ZRQQVUBJGLMDQR
|
7.4 | IC50 | 2 | — | |
RAIVHQQRQQKFFV
|
7.4 | IC50 | 2 | — | |
SYMILEXMAHCATG
|
7.4 | IC50 | 2 | — | |
AYUVNFPAFJUWQW
|
7.3 | IC50 | 2 | — | |
NSNZIHNPWOUVQN
|
7.3 | IC50 | 2 | — | |
NHHQJBCNYHBUSI
|
7.3 | Kd | 220 | — | |
PDMRUTWXKCFDFD
|
7.3 | IC50 | 2 | — | |
CLYZLUAUBTXCPL
|
7.3 | IC50 | 7 | — | |
IWILCSQODDAQDC
|
7.3 | IC50 | 2 | — | |
QTSKVQLIRGIGDV
|
7.3 | IC50 | 3 | — | |
SMAIRFQFHKTXBK
|
7.3 | IC50 | 2 | — | |
PNMCLCQZSVIVDN
|
7.3 | IC50 | 2 | — | |
QMIDZOGAPGBZSC
|
7.3 | IC50 | 4 | — | |
DUUHSIDQKSIHGY
|
7.3 | IC50 | 2 | — | |
KMIUIHAGKAMAMN
|
7.3 | IC50 | 2 | — | |
SINJOIVMLYFADD
|
7.3 | IC50 | 5 | — | |
CIBIQJXLLSSQGJ
|
7.3 | IC50 | 2 | — | |
RDFHITQJRDVSMP
|
7.3 | IC50 | 5 | — | |
RZQANRRMBKDLGQ
|
7.3 | IC50 | 2 | — | |
TUBXJQSNTKADJB
|
7.2 | IC50 | 5 | — | |
ANVBJUPKQASFMW
|
7.2 | IC50 | 3 | — | |
WOTWXKACTZFRQE
|
7.2 | IC50 | 4 | — | |
ZEEVDVUFURMNEH
|
7.2 | IC50 | 2 | — |