Target Details
| UniProt AC | Q9UHD2 |
|---|---|
| Gene Symbol | TBK1 |
| Protein Name | Serine/threonine-protein kinase TBK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18394 (TBK1_CCD1) PF18396 (TBK1_ULD) |
Summary
- Multi-target molecules 639
- Clinical molecules 19
- Avg pChEMBL 7.59
KEGG Pathways (25)
- Alcoholic liver disease
- Amyotrophic lateral sclerosis
- Autophagy - animal
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Pathways of neurodegeneration - multiple diseases
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Shigellosis
- Toll-like receptor signaling pathway
- Yersinia infection
Associated Diseases (3)
Active Molecules (639)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CRYAFKJJVYGHEW
|
7.9 | IC50 | 2 | — | |
HGXOGENWAIQBNI
|
7.8 | IC50 | 2 | — | |
KHKGVBAGOBQZSK
|
7.8 | IC50 | 2 | — | |
LBFKDBMDAOTADZ
|
7.8 | IC50 | 3 | — | |
QQLAYKPAOURFQO
|
7.8 | IC50 | 2 | — | |
SPZBXBBBJTWZTI
|
7.8 | IC50 | 2 | — | |
UXONJEQASGNIRB
|
7.8 | IC50 | 2 | — | |
AKIJKDXIHMPADM
|
7.8 | IC50 | 3 | — | |
BTIIUKSFWMYFNV
|
7.8 | IC50 | 6 | — | |
QQBXPKMQHKPPRH
|
7.8 | IC50 | 3 | — | |
BKJRFMUYVNJZKE
|
7.8 | IC50 | 2 | — | |
YVRJIQLODAYFSS
|
7.8 | IC50 | 2 | — | |
YXLPNLVTKVQNGW
|
7.8 | IC50 | 2 | — | |
HGCJKDOLUCMPFE
|
7.8 | IC50 | 5 | — | |
LHPPCLUNEXZVTH
|
7.8 | IC50 | 2 | — | |
NXSJMRCTGYTSTK
|
7.8 | Kd | 200 | — | |
WEFRCKPVMWDRAK
|
7.8 | IC50 | 5 | — | |
GFHRPONHRZBFNC
|
7.7 | IC50 | 3 | — | |
HNDZOIQVTDQHDZ
|
7.7 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
7.7 | Kd | 289 | Yes | |
UVPLHKWZLRJFSX
|
7.7 | IC50 | 3 | — | |
LZMAOONJSWWBEC
|
7.7 | IC50 | 2 | — | |
UDUUROZQLWGGJD
|
7.7 | IC50 | 2 | — | |
YILMILHQOYYLQQ
|
7.7 | IC50 | 3 | — | |
HNBPCYSNJZUPBY
|
7.7 | IC50 | 2 | — | |
NOCFKKXWSSCWRO
|
7.7 | IC50 | 2 | — | |
SIMRMBMUTPELDR
|
7.7 | IC50 | 2 | — | |
AZBYFLYSUMYTKS
|
7.7 | IC50 | 2 | — | |
IHPBCWXBUXLKAX
|
7.7 | IC50 | 2 | — | |
SQZVSGZHYGZMTP
|
7.7 | IC50 | 2 | — | |
AKBNGGYXMZTHEB
|
7.6 | IC50 | 5 | — | |
VRYICCMNURPSDI
|
7.6 | IC50 | 3 | — | |
WPPGTNKIMPNPSA
|
7.6 | IC50 | 2 | — | |
AEIPIIUQGITKFW
|
7.6 | IC50 | 3 | — | |
HKIHBMOYFPBKRM
|
7.6 | IC50 | 2 | — | |
JASHHRMOVFCTDG
|
7.6 | IC50 | 2 | — | |
JSUQMOCFECZQSH
|
7.6 | IC50 | 2 | — | |
JTBYAWVOSUNWIB
|
7.6 | IC50 | 2 | — | |
KZSBBJDMPIERRN
|
7.6 | IC50 | 2 | — | |
ZGZVRPRSFXRGCF
|
7.6 | Ki | 76 | — | |
RSUXWNMQQLYBIH
|
7.6 | IC50 | 2 | — | |
DYVYNFDWCPVADF
|
7.6 | IC50 | 2 | — | |
DLGOLPMIWUFODI
|
7.6 | IC50 | 2 | — | |
SLCMXEFQPWEZOR
|
7.6 | IC50 | 2 | — | |
KPELCBIAAJVUQI
|
7.5 | IC50 | 3 | — | |
VAVXGGRQQJZYBL
|
7.5 | IC50 | 8 | — | |
JTMNZLVEDRFGHR
|
7.5 | IC50 | 2 | — | |
BGAUWQRNGCAKTK
|
7.5 | IC50 | 2 | — | |
HZRJHVDNTDBTOZ
|
7.5 | IC50 | 8 | — | |
TUIAFUOZECMRAZ
|
7.5 | IC50 | 2 | — |