Target Details
| UniProt AC | Q9UHD2 |
|---|---|
| Gene Symbol | TBK1 |
| Protein Name | Serine/threonine-protein kinase TBK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18394 (TBK1_CCD1) PF18396 (TBK1_ULD) |
Summary
- Multi-target molecules 639
- Clinical molecules 19
- Avg pChEMBL 7.59
KEGG Pathways (25)
- Alcoholic liver disease
- Amyotrophic lateral sclerosis
- Autophagy - animal
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Pathways of neurodegeneration - multiple diseases
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Shigellosis
- Toll-like receptor signaling pathway
- Yersinia infection
Associated Diseases (3)
Active Molecules (639)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WSBKHPYKYJZQTB
|
8.1 | IC50 | 2 | — | |
XKQXMMZJRYXZOV
|
8.1 | IC50 | 3 | — | |
XUCZHDZTLMJKOG
|
8.1 | IC50 | 2 | — | |
YHIJEMUYPDJQLD
|
8.1 | IC50 | 2 | — | |
YIBZCPJGTIQSGV
|
8.1 | IC50 | 2 | — | |
YOFJPZPGHXWQJB
|
8.1 | IC50 | 5 | — | |
ZXXUISVZQNQVSN
|
8.1 | IC50 | 2 | — | |
LNMLTSVLONLVTE
|
8.1 | IC50 | 2 | — | |
AQKBMEOCVCVMRP
|
8.1 | IC50 | 2 | — | |
OSVUGUHRKMMBSE
|
8.1 | Kd | 170 | — | |
PMHQAZQZXRIEPG
|
8.1 | IC50 | 2 | — | |
QELZALHAUCFZNA
|
8.1 | IC50 | 2 | — | |
SNJRVUBJSCKVLN
|
8.1 | IC50 | 5 | — | |
VDDFCDUWOMCJQP
|
8.1 | IC50 | 2 | — | |
WTTGENWPXJVKQI
|
8.1 | IC50 | 3 | — | |
XHNAYNYWJBNROG
|
8.1 | IC50 | 2 | — | |
AXFMFRVMFJMHRE
|
8.0 | IC50 | 2 | — | |
BMGQWWVMWDBQGC
|
8.0 | Kd | 147 | Yes | |
ASPZHEBURRROFC
|
8.0 | IC50 | 2 | — | |
ZNZQEKQKXAOGDX
|
8.0 | IC50 | 2 | — | |
FONLVAFSTIESFR
|
8.0 | IC50 | 2 | — | |
HKVLGLZTELKITJ
|
8.0 | IC50 | 2 | — | |
JUWVGQDRIAVTIK
|
8.0 | IC50 | 3 | — | |
KRCXSXIRZJARBO
|
8.0 | IC50 | 3 | — | |
RSUQGUXLJAJYCT
|
8.0 | IC50 | 2 | — | |
SMBITOOEILSWPI
|
8.0 | IC50 | 2 | — | |
TVLWSLIAVPDZCA
|
8.0 | IC50 | 2 | — | |
VLQLXNFFVREKBK
|
8.0 | IC50 | 3 | — | |
XJXPKTHMXWGQPH
|
8.0 | IC50 | 5 | — | |
FWVWZYYDXODNIY
|
8.0 | IC50 | 2 | — | |
BUHBIIPEWPOROL
|
8.0 | IC50 | 2 | — | |
WTDOVWBIRCFQNH
|
8.0 | IC50 | 3 | — | |
XSPWFBVBJPGXNR
|
8.0 | IC50 | 2 | — | |
HCRPSFHFMMUNAR
|
8.0 | IC50 | 2 | — | |
LUIAXPRIBAAQLN
|
7.9 | IC50 | 2 | — | |
WVQCAVLGAOTNQE
|
7.9 | IC50 | 2 | — | |
FFZYTQWANYSENM
|
7.9 | IC50 | 2 | — | |
OIINJADYHQPDPP
|
7.9 | IC50 | 4 | — | |
RTLHVWFETKCJMG
|
7.9 | IC50 | 3 | — | |
YZWVXQXPLIUUGA
|
7.9 | IC50 | 2 | — | |
ZCCPLJOKGAACRT
|
7.9 | Kd | 599 | — | |
ZNTAAWCMFQAOKC
|
7.9 | IC50 | 3 | — | |
OAYVEVAGVZYBHT
|
7.9 | IC50 | 2 | — | |
WISWDBLLYNYCRE
|
7.9 | IC50 | 2 | — | |
HCQISHRTQSDYMG
|
7.9 | IC50 | 2 | — | |
RYYNGWLOYLRZLK
|
7.9 | Ki | 104 | — | |
IVFSELMCVYLTSD
|
7.9 | IC50 | 3 | — | |
MBYYLRDCKQHUGM
|
7.9 | IC50 | 3 | — | |
JSJHGXYXYWXMNC
|
7.9 | IC50 | 2 | — | |
OESXQVFTYMQBFH
|
7.9 | IC50 | 2 | — |