Target Details
| UniProt AC | Q9UHD2 |
|---|---|
| Gene Symbol | TBK1 |
| Protein Name | Serine/threonine-protein kinase TBK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18394 (TBK1_CCD1) PF18396 (TBK1_ULD) |
Summary
- Multi-target molecules 639
- Clinical molecules 19
- Avg pChEMBL 7.59
KEGG Pathways (25)
- Alcoholic liver disease
- Amyotrophic lateral sclerosis
- Autophagy - animal
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Pathways of neurodegeneration - multiple diseases
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Shigellosis
- Toll-like receptor signaling pathway
- Yersinia infection
Associated Diseases (3)
Active Molecules (639)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SSMPZXRXMBEUFU
|
8.2 | IC50 | 4 | — | |
XNQOGRKQAFZETL
|
8.2 | IC50 | 2 | — | |
AAEIQQDLGQELDQ
|
8.2 | IC50 | 2 | — | |
BCWYUBHSQSCBFH
|
8.2 | IC50 | 2 | — | |
BPNSGZHWOGXFQP
|
8.2 | IC50 | 3 | — | |
CCQLYJZEWHWASR
|
8.2 | IC50 | 5 | — | |
CYCDEYIKBNVSHA
|
8.2 | IC50 | 2 | — | |
DLUFUVCAUGKHRL
|
8.2 | IC50 | 2 | — | |
FNVPRBKVDPEQJB
|
8.2 | IC50 | 3 | — | |
GMCWMRVYPOUFAZ
|
8.2 | IC50 | 2 | — | |
HNLSDFDJZLXTHF
|
8.2 | IC50 | 2 | — | |
JSWSNMUJSFRFCL
|
8.2 | IC50 | 3 | — | |
KICWLQGEPQRPSZ
|
8.2 | IC50 | 3 | — | |
KLRNJRXQJGPXMS
|
8.2 | IC50 | 3 | — | |
KSGXLLJPSWRACC
|
8.2 | IC50 | 2 | — | |
MLQSFEZKSQONMK
|
8.2 | IC50 | 2 | — | |
MQZYHFYFOXLRBV
|
8.2 | IC50 | 2 | — | |
OUYJBEHLMYTWDO
|
8.2 | IC50 | 3 | — | |
PZDIPKRKYNMOJE
|
8.2 | IC50 | 2 | — | |
QLUFGSNYFKCBJT
|
8.2 | IC50 | 3 | — | |
QNAQWEYXUVCFQZ
|
8.2 | IC50 | 3 | — | |
QRQGHALETIKFSZ
|
8.2 | IC50 | 3 | — | |
RVVXQNJZYNFBHM
|
8.2 | IC50 | 3 | — | |
SBZFMUSXXCQCBH
|
8.2 | IC50 | 2 | — | |
TUHJNJJPZVPTPS
|
8.2 | IC50 | 2 | — | |
BGXAJMOKNLNIKN
|
8.2 | IC50 | 2 | — | |
SSFXUEWPQPILFO
|
8.2 | IC50 | 2 | — | |
QZQONLSSIXUDTB
|
8.2 | IC50 | 2 | — | |
UBBGWCKRFYZCTO
|
8.2 | IC50 | 2 | — | |
IVNHCMJOZZBIAP
|
8.2 | IC50 | 2 | — | |
UAROTPQRUDFOGH
|
8.2 | IC50 | 2 | — | |
CIBVSEISWWXHEO
|
8.2 | IC50 | 2 | — | |
CZBLMYRJPRLVRE
|
8.2 | IC50 | 3 | — | |
GCYKYTQSHOSPKE
|
8.2 | IC50 | 3 | — | |
GWPLDWSTEUIHCJ
|
8.2 | IC50 | 3 | — | |
HPLAJCJEPOOJCG
|
8.2 | IC50 | 3 | — | |
MZHPEELZCYWEHG
|
8.2 | IC50 | 6 | — | |
MZKFOXRCMQMVAM
|
8.2 | IC50 | 3 | — | |
PQVPIJFBUFHXCN
|
8.2 | IC50 | 2 | — | |
QVZNMWNIVGLWCE
|
8.2 | IC50 | 2 | — | |
XJRBKRKVNGQEPX
|
8.2 | IC50 | 3 | — | |
ZMKGUWFJWSOBOZ
|
8.1 | IC50 | 2 | — | |
DNGHYRYQEMRIDG
|
8.1 | IC50 | 3 | — | |
IYLJIJFVSGZAIK
|
8.1 | IC50 | 2 | — | |
LFIICVBYLDDKEE
|
8.1 | IC50 | 3 | — | |
NWMPVMMGSHXANZ
|
8.1 | Ki | 58 | — | |
RFPGSBIVMOJECN
|
8.1 | IC50 | 2 | — | |
URECOWLJWSLQCN
|
8.1 | IC50 | 2 | — | |
UUYGOKZIAFBEGX
|
8.1 | IC50 | 3 | — | |
WHHJYUVJNITNFN
|
8.1 | IC50 | 4 | — |