Target Details
| UniProt AC | Q9UHD2 |
|---|---|
| Gene Symbol | TBK1 |
| Protein Name | Serine/threonine-protein kinase TBK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18394 (TBK1_CCD1) PF18396 (TBK1_ULD) |
Summary
- Multi-target molecules 639
- Clinical molecules 19
- Avg pChEMBL 7.59
KEGG Pathways (25)
- Alcoholic liver disease
- Amyotrophic lateral sclerosis
- Autophagy - animal
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Pathways of neurodegeneration - multiple diseases
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Shigellosis
- Toll-like receptor signaling pathway
- Yersinia infection
Associated Diseases (3)
Active Molecules (639)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FKKXZTUVHWKAQM
|
8.4 | IC50 | 3 | — | |
GBDGRXDOLFLBAV
|
8.4 | IC50 | 3 | — | |
GDMLXKZMNHJKNI
|
8.4 | IC50 | 3 | — | |
GWGJYIPISQXQLX
|
8.4 | IC50 | 3 | — | |
HYCRTUWVJJGNKA
|
8.4 | IC50 | 4 | — | |
ICTZCEFKLIZUFV
|
8.4 | IC50 | 3 | — | |
IUDBEIQBJIEKNX
|
8.4 | IC50 | 3 | — | |
KAKYKHXANDESRF
|
8.4 | IC50 | 3 | — | |
LNIQNXFRNKFXIV
|
8.4 | IC50 | 3 | — | |
ORHHPZBLKIDTBX
|
8.4 | IC50 | 3 | — | |
PRELXQNFYRQFTQ
|
8.4 | IC50 | 3 | — | |
VOOUPXYOOCEEFC
|
8.4 | IC50 | 3 | — | |
VZSXBDWSTNVNJE
|
8.4 | IC50 | 2 | — | |
XCYPLUKAXOGVDS
|
8.4 | IC50 | 3 | — | |
XUELBKVSGYWSKD
|
8.4 | IC50 | 4 | — | |
YFBHNTGOTRHQLM
|
8.4 | IC50 | 3 | — | |
ZJRUXNCHFMDOOM
|
8.4 | IC50 | 3 | — | |
ZUUSJSDRSNEYLL
|
8.4 | IC50 | 3 | — | |
JNYUZMNVAQNKRU
|
8.4 | IC50 | 2 | — | |
IOIONYMZILVMCR
|
8.4 | IC50 | 2 | — | |
TXJYLNPKESJZSD
|
8.4 | IC50 | 2 | — | |
XOEXSVADUVFQRN
|
8.4 | IC50 | 2 | — | |
DUEQRTNLBPJYPF
|
8.3 | IC50 | 2 | — | |
ZCTTVOCGTHIYCW
|
8.3 | IC50 | 2 | — | |
BJJXTIWXVHNEJL
|
8.3 | IC50 | 2 | — | |
AYYWOVUIQSBYDE
|
8.3 | IC50 | 3 | — | |
BKPUHGLQZAVNHO
|
8.3 | IC50 | 2 | — | |
CCNUFZSUSDCFGN
|
8.3 | IC50 | 3 | — | |
CMQXQMALEDSQQH
|
8.3 | IC50 | 2 | — | |
DBRHWHXJDUTFKP
|
8.3 | IC50 | 3 | — | |
FJAVKPCYPORWLI
|
8.3 | IC50 | 2 | — | |
FVHKTXLAWSFSNK
|
8.3 | IC50 | 4 | — | |
GCHKGFCTYIRHHF
|
8.3 | IC50 | 3 | — | |
GHMJUVTUHKPGKE
|
8.3 | IC50 | 3 | — | |
IAHBPEPPERDPHA
|
8.3 | IC50 | 2 | — | |
IXEXMSDQIVNECG
|
8.3 | IC50 | 3 | — | |
JSWCKNMMDIGGRJ
|
8.3 | IC50 | 2 | — | |
OFEARPZEWOLQGZ
|
8.3 | IC50 | 4 | — | |
SUGGCBUBUXYRSO
|
8.3 | IC50 | 3 | — | |
SVGGQHQGUDVYQO
|
8.3 | IC50 | 3 | — | |
UONSKTNQTWRUCS
|
8.3 | IC50 | 2 | — | |
VBVBCPLRKQJABM
|
8.3 | IC50 | 3 | — | |
VEMSSQHOLIBJEZ
|
8.3 | IC50 | 3 | — | |
XBFXJAXJSWLRPR
|
8.3 | IC50 | 2 | — | |
FVLDQJNJSJKSKE
|
8.3 | IC50 | 2 | — | |
RNJBPIVRBMZSMD
|
8.3 | IC50 | 2 | — | |
FTVIWWJJRCVHSZ
|
8.3 | IC50 | 2 | — | |
IITKALICJDNWMU
|
8.3 | IC50 | 2 | — | |
MZUYZYAQDFGDQX
|
8.2 | IC50 | 2 | — | |
PERZEHQGYVAHOZ
|
8.2 | IC50 | 2 | — |