Target Details
| UniProt AC | Q9UHD2 |
|---|---|
| Gene Symbol | TBK1 |
| Protein Name | Serine/threonine-protein kinase TBK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18394 (TBK1_CCD1) PF18396 (TBK1_ULD) |
Summary
- Multi-target molecules 639
- Clinical molecules 19
- Avg pChEMBL 7.59
KEGG Pathways (25)
- Alcoholic liver disease
- Amyotrophic lateral sclerosis
- Autophagy - animal
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Pathways of neurodegeneration - multiple diseases
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Shigellosis
- Toll-like receptor signaling pathway
- Yersinia infection
Associated Diseases (3)
Active Molecules (639)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KNCDEVRJJHZTFP
|
8.5 | IC50 | 3 | — | |
KOLYMXQYZQEXIF
|
8.5 | IC50 | 3 | — | |
LRDQYJRVAAGHEK
|
8.5 | IC50 | 3 | — | |
MAGYPARKFHXVPO
|
8.5 | IC50 | 3 | — | |
MGUWFXNRNXEUEB
|
8.5 | IC50 | 3 | — | |
MHRJILLQTVZIBV
|
8.5 | IC50 | 3 | — | |
NKOHMDYLNLLENR
|
8.5 | IC50 | 2 | — | |
NMJIAJITODSLIF
|
8.5 | IC50 | 3 | — | |
OCMXFNGLZPKTFI
|
8.5 | IC50 | 3 | — | |
OYQSRSUSXBDIKK
|
8.5 | IC50 | 3 | — | |
PMQODLVRCODLJS
|
8.5 | IC50 | 3 | — | |
PZTKSZRHTHXHMA
|
8.5 | IC50 | 3 | — | |
SRIFSUWDDPLONW
|
8.5 | IC50 | 3 | — | |
URHODGROVLUHQW
|
8.5 | IC50 | 3 | — | |
VFYVJNXWRBZRHQ
|
8.5 | IC50 | 3 | — | |
VHGHPWKEDSVCPO
|
8.5 | IC50 | 3 | — | |
WUOSUEXRIIWVRA
|
8.5 | IC50 | 3 | — | |
WYPVUHJMFDLNSM
|
8.5 | IC50 | 2 | — | |
XGJGUJSSRHZXEN
|
8.5 | IC50 | 3 | — | |
XWAAZPHGKVWIBO
|
8.5 | IC50 | 3 | — | |
YKBZGTPZXATTES
|
8.5 | IC50 | 3 | — | |
YRMKHJKXKFHXMK
|
8.5 | IC50 | 3 | — | |
YTKXJIKRZSXVIP
|
8.5 | IC50 | 2 | — | |
ZFQFDCSTGATGQP
|
8.5 | IC50 | 4 | — | |
ZXXUISVZQNQVSN
|
8.5 | IC50 | 2 | — | |
ZYIWBKBHSZCDAY
|
8.5 | IC50 | 3 | — | |
GNLWUSMRXGCMEL
|
8.5 | IC50 | 2 | — | |
RFWMIZOXLGRIHV
|
8.5 | IC50 | 2 | — | |
VZLQAULNDFJYPL
|
8.5 | IC50 | 2 | — | |
VMYWSKHQGSIDJS
|
8.5 | IC50 | 2 | — | |
OTDPQDOEHSIHCV
|
8.5 | IC50 | 2 | — | |
HSBRJCXMRYCUJI
|
8.5 | IC50 | 2 | — | |
LDRHKGHHXJWLJD
|
8.5 | IC50 | 2 | — | |
QRICOSSIVLKBBT
|
8.5 | IC50 | 2 | — | |
WPWPOCITVIKSCW
|
8.5 | IC50 | 2 | — | |
WTRFGRRHMCNXPV
|
8.4 | IC50 | 2 | — | |
XKXKAOTUKINWLC
|
8.4 | IC50 | 2 | — | |
OWTXNTZZHGTTPX
|
8.4 | IC50 | 2 | — | |
WKVLVOVZAQKAFP
|
8.4 | IC50 | 2 | — | |
WMGMGJHVTOJFFS
|
8.4 | IC50 | 2 | — | |
MCVZGUNLGAFYGU
|
8.4 | IC50 | 2 | — | |
SBRWSTZGLKCGQC
|
8.4 | IC50 | 2 | — | |
ZKDPTJOJEWYFEP
|
8.4 | IC50 | 2 | — | |
ABJMUSKMRCDMPE
|
8.4 | IC50 | 3 | — | |
BCPZVZDYGYPCDP
|
8.4 | IC50 | 3 | — | |
BTBPQEMNWVDZLK
|
8.4 | IC50 | 2 | — | |
CCLSCLZBGDZBMU
|
8.4 | IC50 | 3 | — | |
CQFQKMKEBSPJGU
|
8.4 | IC50 | 3 | — | |
CYSNREWCZKAVDY
|
8.4 | IC50 | 3 | — | |
DECBFIYBUIMGPR
|
8.4 | IC50 | 3 | — |