Target Details
| UniProt AC | Q9UHD2 |
|---|---|
| Gene Symbol | TBK1 |
| Protein Name | Serine/threonine-protein kinase TBK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18394 (TBK1_CCD1) PF18396 (TBK1_ULD) |
Summary
- Multi-target molecules 639
- Clinical molecules 19
- Avg pChEMBL 7.59
KEGG Pathways (25)
- Alcoholic liver disease
- Amyotrophic lateral sclerosis
- Autophagy - animal
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Pathways of neurodegeneration - multiple diseases
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Shigellosis
- Toll-like receptor signaling pathway
- Yersinia infection
Associated Diseases (3)
Active Molecules (639)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NQLGOSWSXPDDSV
|
8.7 | IC50 | 2 | — | |
NQVRHDTYGKEBDT
|
8.7 | IC50 | 2 | — | |
OOYRAPOOQHGEBB
|
8.7 | IC50 | 3 | — | |
OTUJIVCCULIMCW
|
8.7 | IC50 | 2 | — | |
OWRPZPNMYHZVAB
|
8.7 | IC50 | 2 | — | |
OYQSRSUSXBDIKK
|
8.7 | IC50 | 3 | — | |
QPWPSCNQQGTOFW
|
8.7 | IC50 | 3 | — | |
QUOKNSGMLFDHHY
|
8.7 | IC50 | 3 | — | |
QYECLBIGLCTRAG
|
8.7 | IC50 | 3 | — | |
RTNHWTLGYOUURJ
|
8.7 | IC50 | 2 | — | |
RYQFIFAMXTXXOR
|
8.7 | IC50 | 2 | — | |
SDJZXXAGAUAGTD
|
8.7 | IC50 | 3 | — | |
UVLZXVFRGKXTMK
|
8.7 | IC50 | 2 | — | |
VILUZAYZRGMLRF
|
8.7 | IC50 | 3 | — | |
WRMHBKKOYNOLHH
|
8.7 | IC50 | 2 | — | |
XFQGLEVRHJHNBR
|
8.7 | IC50 | 3 | — | |
XXJDZHFAASXZSR
|
8.7 | IC50 | 2 | — | |
XYLDHWOGWNKCSD
|
8.7 | IC50 | 3 | — | |
YLNRUJJGFNIFJI
|
8.7 | IC50 | 3 | — | |
YPUJLPFDSVVFMZ
|
8.7 | IC50 | 3 | — | |
ZTDINRKSUABPHP
|
8.7 | IC50 | 3 | — | |
PPLYZIXDSCRZFR
|
8.7 | IC50 | 2 | — | |
DTVZKOJSVBWMFX
|
8.7 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
8.7 | IC50 | 408 | — | |
BONUPFNAVKLWCH
|
8.6 | IC50 | 2 | — | |
QMGHHBHPDDAGGO
|
8.6 | IC50 | 2 | — | |
RQMSNFNMLUFOPR
|
8.6 | IC50 | 2 | — | |
CQWNYIBDCMZITR
|
8.6 | IC50 | 2 | — | |
CGDQNIWGTMYVJH
|
8.6 | IC50 | 2 | — | |
CKAWWKPUCRQQGO
|
8.6 | IC50 | 2 | — | |
OKCGDSORGJQEJP
|
8.6 | IC50 | 2 | — | |
YDRISZZAAFDOPR
|
8.6 | IC50 | 2 | — | |
AIDMUEJGKCTNDD
|
8.5 | IC50 | 3 | — | |
CAVHGBLDRHUXIQ
|
8.5 | IC50 | 3 | — | |
CGORDIYPCGPLIZ
|
8.5 | IC50 | 3 | — | |
CMIDPQPFFSHFQU
|
8.5 | IC50 | 3 | — | |
CUIFZDBUFLFELF
|
8.5 | IC50 | 2 | — | |
DPSWJWLFWZHTFD
|
8.5 | IC50 | 3 | — | |
FFTJPMREKVKUKF
|
8.5 | IC50 | 3 | — | |
GFUQWWAFJKBDPB
|
8.5 | IC50 | 3 | — | |
GFUZNXPSFSEACI
|
8.5 | IC50 | 3 | — | |
GHZHOTWEULSCJL
|
8.5 | IC50 | 3 | — | |
GJAQYJWEEXUKPK
|
8.5 | IC50 | 3 | — | |
GJFXOWOMEQKLPP
|
8.5 | IC50 | 3 | — | |
GRPKFQBLNWZZJC
|
8.5 | IC50 | 3 | — | |
HZCTUVOMFAAAFJ
|
8.5 | IC50 | 3 | — | |
IFNASLLOEPLWNG
|
8.5 | IC50 | 3 | — | |
IHWPMUHWLMAGRM
|
8.5 | IC50 | 3 | — | |
ILMIYGFJNQSXMA
|
8.5 | IC50 | 3 | — | |
JOMSKNSFOAKBRO
|
8.5 | IC50 | 3 | — |