Target Details
| UniProt AC | Q9UHD2 |
|---|---|
| Gene Symbol | TBK1 |
| Protein Name | Serine/threonine-protein kinase TBK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18394 (TBK1_CCD1) PF18396 (TBK1_ULD) |
Summary
- Multi-target molecules 639
- Clinical molecules 19
- Avg pChEMBL 7.59
KEGG Pathways (25)
- Alcoholic liver disease
- Amyotrophic lateral sclerosis
- Autophagy - animal
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Pathways of neurodegeneration - multiple diseases
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Shigellosis
- Toll-like receptor signaling pathway
- Yersinia infection
Associated Diseases (3)
Active Molecules (639)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CJQGLUJHMXCLQY
|
6.1 | IC50 | 11 | — | |
KZXWFUQZOSWUCY
|
6.1 | IC50 | 2 | — | |
FLBNLJLONKAPLR
|
6.1 | Kd | 31 | — | |
FQLDODIEEKFQOP
|
6.1 | IC50 | 2 | — | |
WTQDVZNJLFUQDW
|
6.1 | IC50 | 2 | — | |
BWZFHPDMLLCYGG
|
6.1 | IC50 | 2 | — | |
RAXZSEGXMBWYQK
|
6.1 | IC50 | 21 | — | |
CXQHYVUVSFXTMY
|
6.1 | Kd | 154 | — | |
DFMCXVONDDGQIY
|
6.1 | Ki | 66 | — | |
GIWAUMWDROOOBY
|
6.1 | IC50 | 2 | — | |
HJYHJYGXRBYDIG
|
6.1 | Ki | 23 | — | |
OEMAOMXEFJMDSR
|
6.1 | IC50 | 4 | — | |
SEJGTFPOEJWEGG
|
6.1 | Kd | 149 | — | |
XZWVOUQIYLZUCJ
|
6.1 | Ki | 23 | — | |
PMEYAHBGTDHJEZ
|
6.1 | IC50 | 2 | — | |
HIONSSOVORAGDX
|
6.1 | IC50 | 2 | — | |
IVAFRTWUCSWUMI
|
6.1 | IC50 | 2 | — | |
UANVBHMEXMGHSB
|
6.0 | IC50 | 2 | — | |
GIWIOFZXFSKQTE
|
6.0 | IC50 | 4 | — | |
OYONTEXKYJZFHA
|
6.0 | Kd | 69 | Yes | |
ZCBUQCWBWNUWSU
|
6.0 | Kd | 59 | — | |
CJKXRJUXLJTCRE
|
6.0 | IC50 | 3 | — | |
CPOMPMCLFHSOKH
|
6.0 | IC50 | 2 | — | |
DSXDCHYXQFEFIC
|
6.0 | IC50 | 2 | — | |
FBBJGFHGYDVTLK
|
6.0 | IC50 | 3 | — | |
FUMCKNCUEAQHCV
|
6.0 | Ki | 103 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KUMKJWMPOOYVGT
|
6.0 | IC50 | 2 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MDJWRQAHXDUJLV
|
6.0 | IC50 | 3 | — | |
MRUJTDMRVPXECC
|
6.0 | IC50 | 2 | — | |
NHJSUXXVSUKAMS
|
6.0 | IC50 | 2 | — | |
OMWKEJOTYAGCFP
|
6.0 | IC50 | 2 | — | |
QBKUOOQFSVMDPB
|
6.0 | Ki | 31 | — | |
QZLCSJKQXXMWTE
|
6.0 | IC50 | 2 | — | |
RMTFITAOVDYEPI
|
6.0 | IC50 | 2 | — | |
WNPBFIJEFIXYRM
|
6.0 | IC50 | 3 | — | |
ZYXAFPZQDYBFBQ
|
6.0 | IC50 | 3 | — |