Target Details
| UniProt AC | Q9UHD2 |
|---|---|
| Gene Symbol | TBK1 |
| Protein Name | Serine/threonine-protein kinase TBK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF18394 (TBK1_CCD1) PF18396 (TBK1_ULD) |
Summary
- Multi-target molecules 639
- Clinical molecules 19
- Avg pChEMBL 7.59
KEGG Pathways (25)
- Alcoholic liver disease
- Amyotrophic lateral sclerosis
- Autophagy - animal
- Coronavirus disease - COVID-19
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis B
- Hepatitis C
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- IL-17 signaling pathway
- Influenza A
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- Mitophagy - animal
- NOD-like receptor signaling pathway
- Pathways of neurodegeneration - multiple diseases
- RIG-I-like receptor signaling pathway
- Ras signaling pathway
- Shigellosis
- Toll-like receptor signaling pathway
- Yersinia infection
Associated Diseases (3)
Active Molecules (639)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LNIVPTBCCJSTCB
|
9.1 | IC50 | 2 | — | |
NMIDELFSFNCISG
|
9.1 | IC50 | 2 | — | |
XKOFZEQBVZTDKP
|
9.1 | IC50 | 2 | — | |
XZIIRCPKAFVFHW
|
9.1 | IC50 | 2 | — | |
GVXJFRXNNLRSLI
|
9.0 | IC50 | 2 | — | |
LZVZBSNKTPVPEB
|
9.0 | IC50 | 2 | — | |
HXAYGARTNPQTPX
|
9.0 | IC50 | 2 | — | |
NRQATTKRQXGWKI
|
9.0 | IC50 | 2 | — | |
HVZSQXWYDLQJTQ
|
9.0 | IC50 | 2 | — | |
CRTQNZPWVJVSDE
|
9.0 | IC50 | 2 | — | |
DYRXRIMUJAAMQI
|
8.9 | IC50 | 2 | — | |
HSLJCXAGEGDBAU
|
8.9 | IC50 | 2 | — | |
JHCYMEMCUXVAIR
|
8.9 | IC50 | 2 | — | |
ZULNHRNAEOVNJO
|
8.9 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
8.9 | Ki | 118 | — | |
WKOPXZJZJXUFCH
|
8.9 | IC50 | 2 | — | |
CIETZITWMCYAKI
|
8.9 | IC50 | 2 | — | |
WQFRKFJYPSEBPY
|
8.9 | IC50 | 2 | — | |
ABZIEHMTFVZXNY
|
8.9 | IC50 | 2 | — | |
FZHSNZZYHHRLDX
|
8.8 | IC50 | 2 | — | |
SXFYXPVAKZPFNY
|
8.8 | IC50 | 2 | — | |
XSGVWMDUOODJTB
|
8.8 | IC50 | 2 | — | |
HXICXBITQYMWNF
|
8.8 | IC50 | 2 | — | |
PRBYIDLQEMMFNC
|
8.8 | IC50 | 2 | — | |
LDJRWCYJKDXGCY
|
8.8 | IC50 | 2 | — | |
RXRLWNRSQUSJOR
|
8.8 | IC50 | 2 | — | |
BDDBUOVVYOJPSW
|
8.8 | IC50 | 2 | — | |
BMLBSNHUAPOBHI
|
8.8 | IC50 | 2 | — | |
FIISTVNCJUTUKH
|
8.8 | IC50 | 2 | — | |
BXLOFFCDXFSKIE
|
8.8 | IC50 | 2 | — | |
UNZLCMSGBFLOLV
|
8.8 | IC50 | 2 | — | |
RGVXQILQOSLWGS
|
8.7 | IC50 | 2 | — | |
VIURSDPOFRRBCH
|
8.7 | IC50 | 2 | — | |
OYYIEVDIWZMYFO
|
8.7 | IC50 | 2 | — | |
GYXIFIORIDAIKZ
|
8.7 | IC50 | 3 | — | |
AEPJRUANSIXNRU
|
8.7 | IC50 | 3 | — | |
AUVLVGAPOCTIAE
|
8.7 | IC50 | 3 | — | |
BTKYEHNXCFJUHN
|
8.7 | IC50 | 2 | — | |
DFQJNFGZAMXNJM
|
8.7 | IC50 | 3 | — | |
FNPIJCTUNTWVDI
|
8.7 | IC50 | 2 | — | |
FREUQZHGBVWAQT
|
8.7 | IC50 | 2 | — | |
GHZHOTWEULSCJL
|
8.7 | IC50 | 3 | — | |
GXCCDZRRVFNQMR
|
8.7 | IC50 | 3 | — | |
HIAIYCFUWYLWRI
|
8.7 | IC50 | 2 | — | |
IAQRFOBNZQJZEU
|
8.7 | IC50 | 3 | — | |
IQQCLKRZDHVEJC
|
8.7 | IC50 | 3 | — | |
JUSSXPRFOJRUEO
|
8.7 | IC50 | 2 | — | |
LYMQARVHTYDQHO
|
8.7 | IC50 | 2 | — | |
MSXLIUGGWDIIKN
|
8.7 | IC50 | 3 | — | |
NOENZZUCTRZYIH
|
8.7 | IC50 | 3 | — |