Target Details
| UniProt AC | Q9UGN5 |
|---|---|
| Gene Symbol | PARP2 |
| Protein Name | Poly [ADP-ribose] polymerase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00644 (PARP) PF02877 (PARP_reg) PF05406 (WGR) |
Summary
- Multi-target molecules 571
- Clinical molecules 0
- Avg pChEMBL 7.42
KEGG Pathways (2)
Active Molecules (571)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SRPQZLVMAZBVEH
|
8.6 | IC50 | 2 | — | |
HTMPMXJFMOUCOQ
|
8.6 | IC50 | 2 | — | |
LLBQUOHKCAYWBR
|
8.5 | IC50 | 2 | — | |
NANHPXHADBZWEH
|
8.5 | IC50 | 2 | — | |
ORXLIHVWCSCXBW
|
8.5 | IC50 | 2 | — | |
AHIVQGOUBLVTCB
|
8.5 | Ki | 2 | — | |
IOHRTULIGFHGAL
|
8.5 | Ki | 2 | — | |
PXVGNWOIQRDFEX
|
8.5 | IC50 | 2 | — | |
RJIYGYHNEKRSTG
|
8.5 | Ki | 2 | — | |
RJRQJZUWLRXDTF
|
8.5 | Ki | 2 | — | |
WUSATWKNDGXYRU
|
8.5 | IC50 | 2 | — | |
XVWZUMYLDUPVRN
|
8.5 | IC50 | 2 | — | |
JJDFDZDTXGPNIC
|
8.5 | IC50 | 2 | — | |
PGGOMVDSVVGTHN
|
8.5 | IC50 | 2 | — | |
BDGRZWISYNXFKD
|
8.4 | IC50 | 3 | — | |
LIQDGVXNWJAUNO
|
8.4 | IC50 | 6 | — | |
LZMKLHYIPIJTRL
|
8.4 | IC50 | 2 | — | |
XKBLRQOXNMSXTO
|
8.4 | IC50 | 2 | — | |
FMVGMOVFNFTMQG
|
8.4 | IC50 | 2 | — | |
SDQYXOQWRCKNII
|
8.4 | IC50 | 2 | — | |
IULLGBUVNORARL
|
8.4 | Ki | 2 | — | |
LGVIXHMVSRYWJL
|
8.4 | Ki | 2 | — | |
PCHKPVIQAHNQLW
|
8.4 | IC50 | 8 | — | |
UVYVRAATXCFMQQ
|
8.4 | IC50 | 4 | — | |
BSBYIGMCJVUHQV
|
8.4 | IC50 | 2 | — | |
HWGQMRYQVZSGDQ
|
8.4 | IC50 | 6 | — | |
VONMSJQAKXAFNE
|
8.4 | IC50 | 2 | — | |
WJSBPAZKQYZPAE
|
8.4 | IC50 | 2 | — | |
ZGDNFPWQEQSQAA
|
8.4 | IC50 | 3 | — | |
PNRISLRFARDPOP
|
8.4 | IC50 | 2 | — | |
PTRXVEZPOQLFDC
|
8.3 | IC50 | 2 | — | |
CLTQHSPVFLJRRV
|
8.3 | IC50 | 2 | — | |
IADDRMVOCUHETH
|
8.3 | IC50 | 2 | — | |
XQOHUNRPGOTXDR
|
8.3 | IC50 | 3 | — | |
HDFQNQPMGAHQTL
|
8.3 | IC50 | 5 | — | |
DQGBARZZIIDDAZ
|
8.3 | IC50 | 2 | — | |
YNOAURUBJUTHDB
|
8.3 | IC50 | 2 | — | |
KXSIHXHEHABEJX
|
8.3 | Ki | 2 | — | |
LXCLGXFJSUMMJY
|
8.3 | IC50 | 4 | — | |
NUHZJIJDJJVSKK
|
8.3 | IC50 | 3 | — | |
KXXRGTYOVUETBV
|
8.3 | IC50 | 3 | — | |
MSZHRPFWZYCRHL
|
8.3 | IC50 | 2 | — | |
NTYRAXKJQKLKLY
|
8.2 | IC50 | 2 | — | |
CHRQYHKDXOIBPC
|
8.2 | IC50 | 2 | — | |
XKOPYVMSQOJAFI
|
8.2 | IC50 | 2 | — | |
CTLOSZHDGZLOQE
|
8.2 | IC50 | 2 | — | |
PPLKPFGRKQMGRE
|
8.2 | IC50 | 3 | — | |
BIFMDHUVYGGFCU
|
8.2 | IC50 | 10 | — | |
DFAIABHDMOLQDA
|
8.2 | IC50 | 5 | — | |
SBJGLDKVXLKVPI
|
8.2 | IC50 | 2 | — |