Target Details
| UniProt AC | Q9UGN5 |
|---|---|
| Gene Symbol | PARP2 |
| Protein Name | Poly [ADP-ribose] polymerase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00644 (PARP) PF02877 (PARP_reg) PF05406 (WGR) |
Summary
- Multi-target molecules 571
- Clinical molecules 0
- Avg pChEMBL 7.42
KEGG Pathways (2)
Active Molecules (571)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MWIUPFYRAAIUMB
|
9.0 | IC50 | 3 | — | |
NIOMTPKIOLNRTQ
|
9.0 | IC50 | 2 | — | |
RCNMQXVWWXSESA
|
9.0 | IC50 | 3 | — | |
SNSYYJLSJTUZMP
|
9.0 | Ki | 2 | — | |
YNBQAYKYNYRCCA
|
9.0 | IC50 | 2 | — | |
ZDDPBFWHZOJFHF
|
9.0 | IC50 | 6 | — | |
FLCHMGRFSJQORK
|
9.0 | IC50 | 3 | — | |
HMABYWSNWIZPAG
|
9.0 | IC50 | 12 | — | |
WELSPTLZWKCYMB
|
9.0 | IC50 | 3 | — | |
JLVRTMBMCWYGAL
|
8.9 | IC50 | 7 | — | |
WARUZPFHLRLCHE
|
8.9 | IC50 | 7 | — | |
LGFTWORQFUMEPZ
|
8.9 | IC50 | 2 | — | |
TXIZSRVUVVGWCN
|
8.9 | IC50 | 2 | — | |
HTRPLWGQNMXGRD
|
8.9 | IC50 | 3 | — | |
MZLDTLJZDXBQCV
|
8.9 | IC50 | 2 | — | |
PQHSBQMZINJNST
|
8.9 | IC50 | 2 | — | |
DJSXTFVMGSHIQP
|
8.9 | IC50 | 2 | — | |
UPTYBPOYVNYQMT
|
8.9 | IC50 | 7 | — | |
AHIVQGOUBLVTCB
|
8.8 | Ki | 2 | — | |
CDFHCXNQPYQRFI
|
8.8 | IC50 | 2 | — | |
GFUWRTZMZMICED
|
8.8 | IC50 | 3 | — | |
UYSWVENMUWDLDZ
|
8.8 | IC50 | 2 | — | |
DCSUGHIXMFUMOQ
|
8.8 | IC50 | 3 | — | |
JFJGQBKALIOSDA
|
8.8 | IC50 | 3 | — | |
UNIBAROCFQUNJP
|
8.8 | IC50 | 2 | — | |
YCMALEKADPQGHA
|
8.8 | IC50 | 2 | — | |
MLYYYJSVHUVZHH
|
8.8 | IC50 | 3 | — | |
OAFQCDJUMPFXNS
|
8.8 | IC50 | 2 | — | |
IZSILESJFBWTKL
|
8.7 | IC50 | 2 | — | |
CEUSZBDWOAZEBV
|
8.7 | IC50 | 2 | — | |
SJFGTXAAKCLIOI
|
8.7 | IC50 | 2 | — | |
VXXHFHBGNMSWMO
|
8.7 | IC50 | 2 | — | |
GGJVOTFHPYZESL
|
8.7 | IC50 | 4 | — | |
JJCAYWVTBMMQMQ
|
8.7 | IC50 | 2 | — | |
ROBJKLPZIPNAMV
|
8.7 | IC50 | 2 | — | |
GTBYWKYWQWSPTR
|
8.7 | Ki | 2 | — | |
JNAHVYVRKWKWKQ
|
8.7 | Ki | 2 | — | |
JSGRLNJKTKDILH
|
8.7 | Ki | 2 | — | |
MABHSRSWSCMJOM
|
8.7 | IC50 | 2 | — | |
PWESUKOHBQOSBW
|
8.7 | Ki | 2 | — | |
UGDXZOURHPLYNW
|
8.7 | Ki | 2 | — | |
WBSPNPVOFBRUKC
|
8.7 | Ki | 2 | — | |
QYXDDRWHQGGYKR
|
8.7 | IC50 | 2 | — | |
POPCEFBMGMRZJG
|
8.7 | IC50 | 2 | — | |
BJFLQGUKMCVUMZ
|
8.6 | IC50 | 2 | — | |
BWTOWBOMDHKCDB
|
8.6 | IC50 | 7 | — | |
SUFHZCQTMDLDRK
|
8.6 | IC50 | 2 | — | |
VYGPONYCLGMRIN
|
8.6 | IC50 | 2 | — | |
CEABYCITKOLZEE
|
8.6 | IC50 | 4 | — | |
AXXNBSKROWNMJJ
|
8.6 | IC50 | 2 | — |