Target Details
| UniProt AC | Q9UGM1 |
|---|---|
| Gene Symbol | CHRNA9 |
| Protein Name | Neuronal acetylcholine receptor subunit alpha-9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 78
- Clinical molecules 0
- Avg pChEMBL 7.91
KEGG Pathways (2)
Active Molecules (78)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HUFVTTXOVNSUAU
|
7.6 | IC50 | 2 | — | |
ACPHUHSYZGYUCK
|
7.5 | IC50 | 5 | — | |
DRTISZFZZALDJX
|
7.5 | IC50 | 2 | — | |
UFUXIPADWDHAOE
|
7.5 | IC50 | 2 | — | |
HOYQFSSTAMVPMS
|
7.5 | IC50 | 2 | — | |
LSHCDRJBFRVFPC
|
7.5 | IC50 | 3 | — | |
ACPHUHSYZGYUCK
|
7.4 | IC50 | 5 | — | |
VRPFKEQKJXVOEF
|
7.3 | IC50 | 2 | — | |
YXKFMTLNLUJJKO
|
7.2 | IC50 | 3 | — | |
GGHPUTYEGYRSMD
|
7.0 | IC50 | 4 | — | |
PWSZVABQPWCKIQ
|
7.0 | IC50 | 3 | — | |
BCQNEYQXBIQZLI
|
6.9 | IC50 | 2 | — | |
XCCFHIMCLZGLNA
|
6.9 | IC50 | 3 | — | |
HLCVGNISNXRLRJ
|
6.9 | IC50 | 2 | — | |
BYQJMXFDNSVOHH
|
6.8 | IC50 | 2 | — | |
GWMPLPRCVNXVGX
|
6.7 | IC50 | 4 | — | |
ZEGWBRDJSPUKNA
|
6.6 | IC50 | 2 | — | |
ODWWODYTMVKWGE
|
6.5 | IC50 | 5 | — | |
CPIMXZAMIJJWLD
|
6.4 | IC50 | 4 | — | |
DJJSBEHWEBTNKF
|
6.3 | IC50 | 2 | — | |
XLQOVPAFVSHLGV
|
6.3 | IC50 | 2 | — | |
XRRBKIXHRVPVKY
|
6.3 | IC50 | 2 | — | |
FIQKPIGOFVCVTG
|
6.2 | IC50 | 4 | — | |
XFBDKMSGGGCNAI
|
6.2 | IC50 | 11 | — | |
GNYBGWMBQKXKSR
|
6.2 | IC50 | 2 | — | |
NXGWHVWTEAHKPX
|
6.1 | IC50 | 2 | — | |
HFSGGAQSIXRBQM
|
6.0 | IC50 | 2 | — | |
KJQOYUHYAZGPIZ
|
6.0 | IC50 | 2 | — |