Target Details
| UniProt AC | Q9UGM1 |
|---|---|
| Gene Symbol | CHRNA9 |
| Protein Name | Neuronal acetylcholine receptor subunit alpha-9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 78
- Clinical molecules 0
- Avg pChEMBL 7.91
KEGG Pathways (2)
Active Molecules (78)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PREQDDPQCXZODC
|
10.3 | IC50 | 3 | — | |
WKBMTJBSBLBSSP
|
9.6 | IC50 | 2 | — | |
QHPSFIKTRMNNLZ
|
9.5 | IC50 | 2 | — | |
UDWUBMUQFIDTJI
|
9.4 | IC50 | 2 | — | |
PCZIHLUSNJIPJG
|
9.4 | IC50 | 2 | — | |
KJYPAFNUDKVSQB
|
9.4 | IC50 | 2 | — | |
DTXMSRNILWYKMZ
|
9.3 | IC50 | 2 | — | |
LBCONOSZVXIZDN
|
9.3 | IC50 | 2 | — | |
CDNFAKVJGFHDDB
|
9.2 | IC50 | 3 | — | |
UPLKJPLAVVLRRJ
|
9.1 | IC50 | 2 | — | |
MYRZVRHXPAUBQQ
|
8.9 | IC50 | 2 | — | |
VVORNPTYPFGYRF
|
8.8 | IC50 | 2 | — | |
ATSVSZCAZDCSBA
|
8.8 | IC50 | 2 | — | |
HSPAQJZXXJFNJX
|
8.8 | IC50 | 2 | — | |
NXNBLYISDGDSIN
|
8.8 | IC50 | 2 | — | |
VVORNPTYPFGYRF
|
8.8 | IC50 | 2 | — | |
RUEDGHCKLGSDLO
|
8.8 | IC50 | 5 | — | |
IEDFIQCVIQRLBV
|
8.7 | IC50 | 3 | — | |
LBCONOSZVXIZDN
|
8.7 | IC50 | 2 | — | |
QGLFVUPFAKQWIH
|
8.5 | IC50 | 2 | — | |
WESGVHHRAFNWER
|
8.5 | IC50 | 7 | — | |
NGGVRPGLGXDGKP
|
8.5 | IC50 | 7 | — | |
IKBFUAJBNDCGFQ
|
8.5 | IC50 | 7 | — | |
VXJKUKUEMCMGCD
|
8.5 | IC50 | 3 | — | |
TYGGQOXANGOHKM
|
8.4 | IC50 | 3 | — | |
PREQDDPQCXZODC
|
8.4 | IC50 | 2 | — | |
XTMVSVQIYRTKIW
|
8.4 | IC50 | 5 | — | |
AKEWRXXBJJCYIL
|
8.4 | IC50 | 2 | — | |
IXZCXFATJZXLRO
|
8.3 | IC50 | 3 | — | |
MAZBMPSWUMNOSJ
|
8.3 | IC50 | 3 | — | |
IUEKLDYMAHZDFO
|
8.3 | IC50 | 3 | — | |
VFBLBKKMLKAPON
|
8.3 | IC50 | 2 | — | |
GLILJDHGIUHYHF
|
8.3 | IC50 | 3 | — | |
SYHUNRXHLPKXCV
|
8.2 | IC50 | 2 | — | |
ZSABOEGCGSSQQO
|
8.2 | IC50 | 2 | — | |
BZGYSFMJVCMPRM
|
8.2 | IC50 | 3 | — | |
JRAZMHFHZFKHQJ
|
8.2 | IC50 | 7 | — | |
MFZDCTGKYAGWRM
|
8.2 | IC50 | 3 | — | |
YIMFXBPXUPTIEJ
|
8.0 | IC50 | 7 | — | |
ILEWLUJOKLLBMF
|
8.0 | IC50 | 7 | — | |
QSZLRCIREBTJEI
|
8.0 | IC50 | 2 | — | |
ZGMXUPVWRQVUKG
|
7.9 | IC50 | 4 | — | |
JJGCCLFTIIFXFM
|
7.9 | IC50 | 3 | — | |
KVAQWDSPULTKDL
|
7.8 | IC50 | 2 | — | |
LTQVQLWABHPOHE
|
7.8 | IC50 | 2 | — | |
TVHOLQCXRVTWBY
|
7.8 | IC50 | 4 | — | |
WQOBFWQJRGVMQX
|
7.8 | IC50 | 5 | — | |
KZTLNPPLLLJLHU
|
7.8 | IC50 | 7 | — | |
VVDRDHLUVVGURR
|
7.7 | IC50 | 5 | — | |
CMYORFAIGQYXOW
|
7.7 | IC50 | 2 | — |