Target Details
| UniProt AC | Q9UGI9 |
|---|---|
| Gene Symbol | PRKAG3 |
| Protein Name | 5'-AMP-activated protein kinase subunit gamma-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00571 (CBS) |
Summary
- Multi-target molecules 30
- Clinical molecules 5
- Avg pChEMBL 7.14
KEGG Pathways (16)
- AMPK signaling pathway
- Adipocytokine signaling pathway
- Alcoholic liver disease
- Apelin signaling pathway
- Circadian rhythm
- FoxO signaling pathway
- Glucagon signaling pathway
- Hypertrophic cardiomyopathy
- Insulin resistance
- Insulin signaling pathway
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- Non-alcoholic fatty liver disease
- Oxytocin signaling pathway
- Thermogenesis
- Tight junction
Active Molecules (30)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FJNHSBVZTQFKEF
|
9.0 | IC50 | 7 | — | |
JKGJLUCJLNJXKG
|
8.6 | IC50 | 7 | — | |
FCLPVPNWFDOVKL
|
8.4 | Ki | 11 | — | |
NOMBUNHXDWBICV
|
8.3 | Ki | 11 | — | |
CXYVYGXMFQSTKH
|
8.2 | IC50 | 7 | — | |
XRDMDDSSWUSOAX
|
8.1 | IC50 | 7 | — | |
WGWCRXQUBYJTRA
|
8.0 | Ki | 11 | — | |
WQUGCKCCOOBUNT
|
7.8 | IC50 | 7 | — | |
QZCUYXGDXFPQEA
|
7.7 | IC50 | 7 | — | |
NTZCHZCFSJZAQG
|
7.7 | IC50 | 7 | — | |
MRMDURIHTGUZQI
|
7.5 | IC50 | 7 | — | |
OFPXCBKYWWZZGT
|
7.2 | IC50 | 7 | — | |
WMXDIPVFXWNELM
|
7.2 | IC50 | 14 | Yes | |
XHBVYDAKJHETMP
|
7.0 | IC50 | 24 | Yes | |
BPMMMRKHRUQAAY
|
6.9 | IC50 | 7 | — | |
JRKYKAKARRYSSS
|
6.8 | IC50 | 14 | Yes | |
UDMBCSSLTHHNCD
|
6.8 | Kd | 11 | — | |
LLRSNVNZYTWKPN
|
6.7 | IC50 | 7 | — | |
IUDLPZTURGVXEA
|
6.7 | Kd | 7 | — | |
HEPDAJRNJBNJAE
|
6.7 | IC50 | 15 | Yes | |
PIVGOZQUWKCUID
|
6.6 | IC50 | 7 | — | |
VCLMLPXAUIQEEM
|
6.6 | IC50 | 7 | — | |
OOQJIJYKWXLQNC
|
6.5 | IC50 | 16 | Yes | |
ZXOKHOODFVNZIC
|
6.3 | IC50 | 7 | — | |
CQZOSLVFDRPCFJ
|
6.3 | IC50 | 7 | — | |
WNLKAYDTKKISBN
|
6.2 | IC50 | 7 | — | |
INGGFDWTZNSBPY
|
6.1 | IC50 | 7 | — | |
NGDYCJGYGAYDIM
|
6.1 | IC50 | 7 | — | |
ZWIGVNWZHBPXNS
|
6.1 | IC50 | 7 | — | |
BUMYTKZYNNGHLL
|
6.0 | IC50 | 7 | — |