Target Details
| UniProt AC | Q9UF33 |
|---|---|
| Gene Symbol | EPHA6 |
| Protein Name | Ephrin type-A receptor 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF07699 (Ephrin_rec_like) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 32
- Clinical molecules 17
- Avg pChEMBL 6.74
KEGG Pathways (1)
Active Molecules (32)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CXQHYVUVSFXTMY
|
9.0 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
8.8 | Kd | 149 | — | |
WVXNSAVVKYZVOE
|
7.8 | IC50 | 92 | — | |
SFCBIFOAGRZJNX
|
7.7 | Kd | 22 | — | |
XXJWYDDUDKYVKI
|
7.4 | Kd | 52 | — | |
UHTHHESEBZOYNR
|
7.3 | Kd | 66 | Yes | |
KTEIFNKAUNYNJU
|
7.2 | Kd | 114 | — | |
VAARYSWULJUGST
|
7.2 | Kd | 119 | Yes | |
NHHQJBCNYHBUSI
|
6.9 | Kd | 220 | — | |
QQWUGDVOUVUTOY
|
6.9 | Kd | 231 | Yes | |
WCWUXEGQKLTGDX
|
6.7 | Kd | 22 | Yes | |
MFAQYJIYDMLAIM
|
6.7 | Kd | 130 | Yes | |
UIARLYUEJFELEN
|
6.6 | Kd | 289 | Yes | |
HKSZLNNOFSGOKW
|
6.6 | Kd | 408 | — | |
ZCCPLJOKGAACRT
|
6.6 | IC50 | 599 | — | |
OMZCMEYTWSXEPZ
|
6.6 | Kd | 43 | Yes | |
MPVGZUGXCQEXTM
|
6.5 | Kd | 61 | Yes | |
ULXXDDBFHOBEHA
|
6.5 | Kd | 15 | Yes | |
MLDQJTXFUGDVEO
|
6.4 | Kd | 85 | Yes | |
ODPGGGTTYSGTGO
|
6.4 | Kd | 153 | — | |
YYLKKYCXAOBSRM
|
6.4 | Kd | 191 | — | |
MVCOAUNKQVWQHZ
|
6.4 | Kd | 54 | Yes | |
RAHBGWKEPAQNFF
|
6.3 | Kd | 26 | — | |
HHFBDROWDBDFBR
|
6.2 | Kd | 40 | Yes | |
XGALLCVXEZPNRQ
|
6.2 | Kd | 39 | Yes | |
AAKJLRGGTJKAMG
|
6.2 | Kd | 50 | Yes | |
HHZIURLSWUIHRB
|
6.2 | Kd | 57 | Yes | |
XZXHXSATPCNXJR
|
6.0 | Kd | 165 | Yes | |
WINHZLLDWRZWRT
|
6.0 | Kd | 201 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |