Target Details
| UniProt AC | Q9UEW8 |
|---|---|
| Gene Symbol | STK39 |
| Protein Name | STE20/SPS1-related proline-alanine-rich protein kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF12202 (OSR1_C) PF00069 (Pkinase) |
Summary
- Multi-target molecules 10
- Clinical molecules 4
- Avg pChEMBL 6.59
KEGG Pathways (1)
Active Molecules (10)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
7.8 | IC50 | 408 | — | |
IEDDDZFQZKDRBJ
|
7.5 | IC50 | 9 | — | |
WINHZLLDWRZWRT
|
6.8 | Kd | 201 | Yes | |
QQWUGDVOUVUTOY
|
6.8 | Kd | 231 | Yes | |
CTNPALGJUAXMMC
|
6.4 | Kd | 151 | — | |
PIQCTGMSNWUMAF
|
6.3 | Kd | 137 | Yes | |
XZXHXSATPCNXJR
|
6.3 | Kd | 165 | Yes | |
YYLKKYCXAOBSRM
|
6.0 | Kd | 191 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |