Target Details
| UniProt AC | Q9UEE5 |
|---|---|
| Gene Symbol | STK17A |
| Protein Name | Serine/threonine-protein kinase 17A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 277
- Clinical molecules 13
- Avg pChEMBL 6.99
Active Molecules (277)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YUOWJICKAJQZLS
|
6.2 | Ki | 35 | — | |
UZWDCWONPYILKI
|
6.2 | IC50 | 47 | — | |
AXRCEOKUDYDWLF
|
6.1 | Kd | 31 | — | |
ATVTUVKVZSYFBE
|
6.1 | IC50 | 7 | — | |
CALAEFSQWBJMDU
|
6.1 | Ki | 21 | — | |
GHAZVJQMLWOQLP
|
6.1 | Ki | 17 | — | |
GQGMUKOYILWOIQ
|
6.1 | Ki | 25 | — | |
JZTOUVBEZONDKA
|
6.1 | Ki | 80 | — | |
NEWAULHLLUCDPD
|
6.1 | Ki | 27 | — | |
OEKYVFZKBRIDJO
|
6.1 | Ki | 12 | — | |
RGOPHVZLEMGMBZ
|
6.1 | Ki | 20 | — | |
WINHZLLDWRZWRT
|
6.1 | Ki | 66 | — | |
WPHKIQPVPYJNAX
|
6.1 | Ki | 81 | — | |
WYLVFMBGPRCDQF
|
6.1 | Ki | 14 | — | |
XPHWIERLJBFPFV
|
6.1 | Ki | 69 | — | |
PIQCTGMSNWUMAF
|
6.1 | Kd | 137 | Yes | |
CLEGDJQQHUTCOW
|
6.0 | Ki | 43 | — | |
CPGKMMMSMJKHDL
|
6.0 | Ki | 16 | — | |
FGLPGUCHBHILNS
|
6.0 | Ki | 10 | — | |
IFPPYSWJNWHOLQ
|
6.0 | Ki | 52 | Yes | |
KAICHBSRWFIESE
|
6.0 | Ki | 14 | — | |
KVYKDXMRLMPSGQ
|
6.0 | Ki | 7 | — | |
OEEGUWWPGAZRIJ
|
6.0 | Ki | 21 | — | |
PAIFYAZSILXLBO
|
6.0 | Ki | 26 | — | |
RTDSHUGNRVXRHN
|
6.0 | Ki | 51 | — | |
ZDXCUVXIHVTLEU
|
6.0 | Ki | 3 | — | |
ZGDSBEUMPIMXBM
|
6.0 | Ki | 42 | — |