Target Details
UniProt ACQ9UEE5
Gene SymbolSTK17A
Protein NameSerine/threonine-protein kinase 17A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00069 (Pkinase)
Summary
  • Multi-target molecules 277
  • Clinical molecules 13
  • Avg pChEMBL 6.99
Top Co-occurrence Targets
Active Molecules (277)
InChIKey pChEMBL Type Targets Clinical
PKEYNQACQWYICF 6.5 IC50 6
JWNPDZNEKVCWMY 6.5 Kd 57 Yes
JGIGRRQUXCRVAK 6.4 IC50 2
OSVUGUHRKMMBSE 6.4 Kd 170
PKYSCANLQNSBRH 6.4 IC50 2
BBZSEXSOPOXLIQ 6.4 Ki 8
CACMTVGXYAZZNY 6.4 Ki 11
CHTMRWQLNNRRFJ 6.4 Ki 70
CNQGNADBGYCKKV 6.4 Ki 25
DBXGGXLBTWZXBB 6.4 Ki 39
OADRBDVURCEKRP 6.4 Ki 44
PCQMERRARZKTPW 6.4 Ki 68
PNAPQQCRNHMIER 6.4 Ki 12
SGHXFHRRWFLILP 6.4 Ki 29
SJDGHXXYFFXVPE 6.4 Ki 9
UXUQVXDYXKMCGA 6.4 Ki 21
XSDJOIOVIMPMHD 6.4 Ki 44
YGUMGYOBTNGZKS 6.4 Ki 12
ZRQXCQXWTLVASO 6.4 Ki 36
MHPBLCYPFBBOND 6.4 IC50 6
BNYXRPMABDQJJR 6.4 Kd 5
NXWXUDHOUKWAQU 6.4 Kd 16
OUSFTKFNBAZUKL 6.4 Kd 58 Yes
UVLOISNMRLZTPF 6.4 IC50 5
WXRNDKRLCQNQGX 6.3 IC50 2
BLTVBQXJFVRPFK 6.3 Ki 7
DJUSDFVEBBYFFL 6.3 Ki 27
GNZPMJDEUIVORU 6.3 Ki 3
GQHMZZXJWGPHDA 6.3 Ki 20
HRJWTAWVFDCTGO 6.3 Ki 13 Yes
IMMZLRQJNZSTTE 6.3 Ki 15
ISEDKXOMRIKZPK 6.3 Ki 13
JOIUJUJSHIHBDT 6.3 Ki 18
NJPWCTYVEJIQBM 6.3 Ki 72
UMTWTCVTRDYHQQ 6.3 Ki 56
VQPBIJGXSXEOCU 6.3 Ki 24
YKJSWMAVAKRUAN 6.3 Ki 19
ZVZCNOQSOULQEK 6.3 Ki 2
JOOXLOJCABQBSG 6.2 Kd 139
GDYZFFBMSBDTAA 6.2 Ki 60
GLMWKEAUVZDGKE 6.2 Ki 23
HGVYGHNZFIZVJT 6.2 IC50 2
IJRBJCMLWLFMIN 6.2 Ki 17
IOYFYUOBKSQTFF 6.2 IC50 3
KNVOICXEDILAGT 6.2 Ki 17
MQAKXLBEDXFDMV 6.2 Ki 5
OUJZYQBEFNDJQN 6.2 Ki 71
SKKRZILJUKYLJS 6.2 Ki 25
SQXSMLLCDWJNAC 6.2 Ki 20
VXYDJXMHISGSDA 6.2 Ki 59
2D structure