Target Details
| UniProt AC | Q9UEE5 |
|---|---|
| Gene Symbol | STK17A |
| Protein Name | Serine/threonine-protein kinase 17A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 277
- Clinical molecules 13
- Avg pChEMBL 6.99
Active Molecules (277)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZGGIYFOLDBTZIL
|
7.3 | Ki | 27 | — | |
ZGZVRPRSFXRGCF
|
7.3 | Ki | 76 | — | |
QSDUMEKQISKWQM
|
7.3 | IC50 | 2 | — | |
YQKQQLKFPBCSDP
|
7.2 | IC50 | 2 | — | |
OJBZKMRHGQTLHT
|
7.2 | IC50 | 2 | — | |
AOBLBPWPSKBHSI
|
7.2 | Ki | 55 | — | |
DKXHSOUZPMHNIZ
|
7.2 | Ki | 51 | Yes | |
DQPYZHUAILXFJI
|
7.2 | Ki | 27 | — | |
GQLWKGVBOIYMTN
|
7.2 | Ki | 35 | — | |
HOYRWTWZUFFACV
|
7.2 | Ki | 28 | — | |
KJVWCDAPVMWKLJ
|
7.2 | Ki | 20 | — | |
OWFLADWRSCINST
|
7.2 | Ki | 30 | — | |
SMRWVXLSRJWVBF
|
7.2 | Ki | 25 | — | |
RSZNIJJWHYKJKS
|
7.2 | IC50 | 2 | — | |
CMWRPDHVGMHLSZ
|
7.2 | IC50 | 22 | — | |
DFMCXVONDDGQIY
|
7.1 | Ki | 66 | — | |
HEUSUIRCBWROMH
|
7.1 | Ki | 64 | — | |
LPILBMJJRGTKOQ
|
7.1 | Ki | 27 | — | |
QATMNAAQTUISJK
|
7.1 | Ki | 13 | — | |
QNUKRWAIZMBVCU
|
7.1 | Ki | 46 | — | |
SBFPHSVZEXSHTL
|
7.1 | Ki | 62 | — | |
SRONQUHCRFZABC
|
7.1 | Ki | 28 | — | |
YKYRQCWLYUTVIE
|
7.1 | Ki | 16 | — | |
QKAONCSNINNEGU
|
7.0 | Kd | 5 | — | |
IQNOGQGSOHNMCL
|
7.0 | Ki | 14 | — | |
KYACBMRLQMEIAI
|
7.0 | Ki | 30 | — | |
MJWLCXWVFUXXNZ
|
7.0 | Kd | 3 | — | |
OWRXHGAFWZFFCW
|
7.0 | Ki | 113 | — | |
PQOAVBVTXNJMCM
|
7.0 | Ki | 8 | — | |
ZUKXESAZGMJHLJ
|
7.0 | IC50 | 4 | — | |
CZBQLMXEBSGXMK
|
7.0 | IC50 | 2 | — | |
XZXHXSATPCNXJR
|
7.0 | Kd | 165 | Yes | |
HDAJDNHIBCDLQF
|
6.9 | IC50 | 14 | — | |
LIMMMAWLSIHXGX
|
6.9 | IC50 | 5 | — | |
VVFCWFGNLTVHBL
|
6.9 | IC50 | 5 | — | |
CZIGMBNEFWBEMD
|
6.9 | Ki | 16 | — | |
DBKQWGCVGCVPIP
|
6.9 | Ki | 21 | — | |
IABDKYMGRMDGMM
|
6.9 | Ki | 10 | — | |
KAZJIBCOYQRDGG
|
6.9 | Ki | 16 | — | |
NXNQLECPAXXYTR
|
6.9 | Ki | 29 | — | |
PJLYZTYJSMPZHT
|
6.9 | IC50 | 2 | — | |
SLKCVFPEQGHNSI
|
6.9 | Ki | 29 | — | |
UMYBAQLXZPEUQW
|
6.9 | Ki | 15 | — | |
VIJBEUTVNBPGIU
|
6.9 | Ki | 19 | — | |
WUWDLXZGHZSWQZ
|
6.9 | Ki | 41 | — | |
XUFLBSMTYMFOQH
|
6.9 | Ki | 43 | — | |
YWTBGJGMTBHQTM
|
6.9 | Ki | 65 | — | |
ZKHDDJKHTPLPOQ
|
6.9 | Ki | 62 | — | |
HKTBYUWLRDZAJK
|
6.9 | IC50 | 5 | — | |
DYSRECIVMDGUQU
|
6.8 | Ki | 29 | — |