Target Details
| UniProt AC | Q9UEE5 |
|---|---|
| Gene Symbol | STK17A |
| Protein Name | Serine/threonine-protein kinase 17A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 277
- Clinical molecules 13
- Avg pChEMBL 6.99
Active Molecules (277)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ATWJOSDBVRWRHS
|
7.6 | IC50 | 5 | — | |
CUGHJABOPLILMY
|
7.6 | IC50 | 2 | — | |
NMTICOSWEFXQCN
|
7.6 | IC50 | 2 | — | |
CTNPALGJUAXMMC
|
7.6 | Kd | 151 | — | |
FNCKZBZRSNSOLA
|
7.6 | IC50 | 2 | — | |
HRSFSLVREYGRTM
|
7.6 | IC50 | 2 | — | |
LPTRUOTUVXADBL
|
7.6 | IC50 | 2 | — | |
OFYQAVFEGWZUOW
|
7.6 | IC50 | 2 | — | |
ACSYKUPGCXYRRO
|
7.6 | Ki | 26 | — | |
MDJCUXFFMNEBHG
|
7.6 | Ki | 13 | — | |
RKUKAACYUCUJEE
|
7.6 | Ki | 58 | — | |
XJXPKTHMXWGQPH
|
7.6 | IC50 | 5 | — | |
YMIJUBCSOKSFRU
|
7.6 | Ki | 87 | — | |
HKSZLNNOFSGOKW
|
7.6 | IC50 | 408 | — | |
RXEFTAHHUZTOCL
|
7.6 | IC50 | 2 | — | |
UUSZNXFMBUWTTJ
|
7.6 | IC50 | 2 | — | |
CTMGXPGMEMDNLR
|
7.6 | IC50 | 2 | — | |
MZHPEELZCYWEHG
|
7.5 | IC50 | 6 | — | |
ADMFLILDQJSEIK
|
7.5 | Ki | 72 | — | |
BGYVWFZMYBWCNY
|
7.5 | Ki | 30 | — | |
DTMZXHDQZQLTHA
|
7.5 | Ki | 21 | — | |
JJTYLBBKGQOISV
|
7.5 | Ki | 15 | — | |
LRINYHMQZRENCY
|
7.5 | Ki | 29 | — | |
OLVBAUVSICCWEJ
|
7.5 | Ki | 39 | — | |
PLHUMPJXRHMFFR
|
7.5 | Ki | 28 | — | |
QVJYGMLAIWRCFT
|
7.5 | IC50 | 5 | — | |
WDARYLSSWBWVCU
|
7.5 | Ki | 49 | — | |
YEHCNYAQEBQCCS
|
7.5 | Ki | 74 | — | |
ZLVOTRRGLSDLPF
|
7.5 | Ki | 36 | — | |
NHHQJBCNYHBUSI
|
7.5 | Kd | 220 | — | |
YCFFONJEHNSECY
|
7.5 | IC50 | 2 | — | |
KLKGPGDTGWFQGS
|
7.5 | IC50 | 2 | — | |
MJPLWOKXLCUJOE
|
7.5 | IC50 | 2 | — | |
RVPBVWKXJFMDLI
|
7.5 | IC50 | 2 | — | |
GBHDESSDDILIEU
|
7.4 | IC50 | 2 | — | |
RTXOFPOQIUYKBR
|
7.4 | IC50 | 2 | — | |
CYLGCMABIBXHIQ
|
7.4 | Ki | 16 | — | |
FUMCKNCUEAQHCV
|
7.4 | Ki | 103 | — | |
GCBJDOWIQHMCMR
|
7.4 | Ki | 84 | — | |
HSMUWLLZAZCLHF
|
7.4 | Ki | 25 | — | |
IUEBPIPDFMCSTP
|
7.4 | Ki | 29 | — | |
KRIUNPBAQZGFQA
|
7.4 | Ki | 76 | — | |
LRZYYIZFBXFSJB
|
7.4 | Ki | 69 | — | |
LYNBNVBMAGDJRW
|
7.4 | Ki | 81 | — | |
UQJQNZHGEVLHST
|
7.4 | Ki | 15 | — | |
UKBGBACORPRCGG
|
7.4 | IC50 | 17 | — | |
BMTCUOGIUBLWDI
|
7.4 | IC50 | 2 | — | |
GXYHQFWLVGXTTH
|
7.3 | IC50 | 2 | — | |
FAUVGWZEHNGPFI
|
7.3 | IC50 | 3 | — | |
NHFDRBXTEDBWCZ
|
7.3 | Ki | 41 | — |